| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4202136 | B | Displacement of [3H]reserpine from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 2. | ALA4202137 | B | Displacement of [3H]DHTB from human VMAT2 expressed in HEK293 cell membranes incubated for 90 mins by microbeta scintillation counting method | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 3. | ALA4202144 | B | Displacement of [3H](+)-syn-Ethyl 1-(2-(2,4-Dioxo-1,2-dihydroquinazolin-3(4H)-yl)ethyl)-4-(4-fluorophenyl)piperidine-3-carboxylate from human VMAT2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 4. | ALA4202145 | B | Inhibition of human VMAT2 expressed in HEK293 cell membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addition and measured after 6 mins | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 5. | ALA4202146 | B | Inhibition of VMAT2 in C57Bl/6J mouse striatal membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addition and measured after 8 mins | Mus musculus | 19 | cell membrane format | Scientific Literature | ||
| 6. | ALA4202147 | B | Displacement of [125I]DOI from human 5HT2A receptor expressed in HEK293 cell membranes | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 7. | ALA4202148 | B | Displacement of [125I]RTI-55 from human DAT expressed in HEK293 cell membranes | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 8. | ALA4202149 | B | Displacement of [125I]RTI-55 from human SERT expressed in HEK293 cell membranes | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 9. | ALA4202150 | B | Displacement of [125I]RTI-55 from human NET expressed in HEK293 cell membranes | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 10. | ALA4202151 | B | Binding affinity to 5HT1A receptor (unknown origin) | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 11. | ALA4202152 | A | Cytotoxicity in HEK293 cells expressing human VMAT2 assessed as reduction in cell viability at 10 uM incubated for 24 hrs by MTT assay | Homo sapiens | 10 | cell-based format | Scientific Literature |
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