| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4200085 | F | Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay | Homo sapiens | 51 | cell-based format | Scientific Literature | ||
| 2. | ALA4200086 | F | Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay relative to MDL 29,951 | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
| 3. | ALA4200095 | F | Agonist activity at rat GPR17 expressed in HEK293 cells assessed as induction of intracellular calcium mobilization by calcium 5-dye based assay | Rattus norvegicus | 3 | cell-based format | Scientific Literature | ||
| 4. | ALA4200096 | F | Agonist activity at mouse GPR17 expressed in HEK293 cells assessed as induction of intracellular calcium mobilization by calcium 5-dye based assay | Mus musculus | 3 | cell-based format | Scientific Literature | ||
| 5. | ALA4200097 | F | Agonist activity at rat GPR17 expressed in HEK293 cells assessed as induction of intracellular calcium mobilization at 10 uM by calcium 5-dye based assay relative to MDL 29,951 | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA4200098 | F | Agonist activity at mouse GPR17 expressed in HEK293 cells assessed as induction of intracellular calcium mobilization at 10 uM by calcium 5-dye based assay relative to MDL 29,951 | Mus musculus | 2 | cell-based format | Scientific Literature | ||
| 7. | ALA4200099 | F | Agonist activity at human P2Y1 receptor transfected in human 1321N1 cells assessed as induction of calcium mobilization after 30 mins in presence of ADP by fluo-4 dye based assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 8. | ALA4200100 | F | Agonist activity at human P2Y2 receptor transfected in human 1321N1 cells assessed as induction of calcium mobilization after 30 mins in presence of UTP by fluo-4 dye based assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 9. | ALA4200101 | F | Agonist activity at human P2Y4 receptor transfected in human 1321N1 cells assessed as induction of calcium mobilization after 30 mins in presence of UTP by fluo-4 dye based assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 10. | ALA4200102 | F | Agonist activity at human P2Y6 receptor transfected in human 1321N1 cells assessed as induction of calcium mobilization after 30 mins in presence of UDP by fluo-4 dye based assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 11. | ALA4200103 | F | Agonist activity at human P2Y12 receptor transfected in CHO cells assessed as induction of beta-arrestin translocation | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 12. | ALA4200104 | F | Agonist activity at human P2Y14 receptor transfected in CHO cells assessed as induction of beta-arrestin translocation | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 13. | ALA4200106 | B | Selectivity ratio of EC50 for rat GPR17 expressed in HEK293 cells to EC50 for human GPR17 expressed in human 1321N1 cells | 3 | cell-based format | Scientific Literature | |||
| 14. | ALA4200107 | B | Selectivity ratio of EC50 for mouse GPR17 expressed in HEK293 cells to EC50 for human GPR17 expressed in human 1321N1 cells | 3 | cell-based format | Scientific Literature | |||
| 15. | ALA4200108 | B | Displacement of [3H]PSB-12150 from human GPR17 expressed in CHO cell membranes after 60 mins by liquid scintillation counting | Homo sapiens | 3 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!