| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4190620 | Binding | Inhibition of GABA-A (unknown origin) | Homo sapiens | 1 | ALA4190175 | assay format | Scientific Literature | |
| 2. | ALA4190621 | Binding | Antagonist activity at human TRPA1 oS5 chimera containing (870 to 896 residues) expressed in 293-T-REx cells at holding potential of 15 mV measured after 1 min by PatchXpress electrophysiology assay | Homo sapiens | 1 | ALA4190175 | cell-based format | Scientific Literature | |
| 3. | ALA4190622 | ADME | Stability in human liver microsomes assessed as metabolic turnover number at 10 uM after 15 mins by LC-MS/UV analysis | Homo sapiens | 32 | ALA4190175 | microsome format | Scientific Literature | |
| 4. | ALA4190623 | ADME | Passive permeability of the compound in RRCK cells | Canis lupus familiaris | 32 | ALA4190175 | cell-based format | Scientific Literature | |
| 5. | ALA4190625 | Physicochemical | Lipophilicity, log D of the compound | 2 | ALA4190175 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA4190626 | ADME | Ratio of permeability from basolateral to apical side over apical to basolateral side in RRCK cells expressing MDR1 | Canis lupus familiaris | 2 | ALA4190175 | cell-based format | Scientific Literature | |
| 7. | ALA4190627 | Physicochemical | Dissociation constant, pKa of the compound | 1 | ALA4190175 | small-molecule physicochemical format | Scientific Literature | ||
| 8. | ALA4190628 | Binding | Antagonist activity at human TRPA1 by electrophysiology assay | Homo sapiens | 1 | ALA4190175 | single protein format | Scientific Literature | |
| 9. | ALA4190629 | Binding | Antagonist activity at rat TRPA1 by electrophysiology assay | Rattus norvegicus | 2 | ALA4190175 | single protein format | Scientific Literature | |
| 10. | ALA4190630 | Binding | Antagonist activity at mouse TRPA1 by electrophysiology assay | Mus musculus | 1 | ALA4190175 | single protein format | Scientific Literature | |
| 11. | ALA4190631 | Binding | Antagonist activity at pig TRPA1 by electrophysiology assay | Sus scrofa | 1 | ALA4190175 | assay format | Scientific Literature | |
| 12. | ALA4190632 | ADME | Stability in human hepatocytes | Homo sapiens | 1 | ALA4190175 | cell-based format | Scientific Literature | |
| 13. | ALA4190633 | ADME | Stability in rat liver microsomes | Rattus norvegicus | 1 | ALA4190175 | microsome format | Scientific Literature | |
| 14. | ALA4190634 | ADME | Stability in rat hepatocytes | Rattus norvegicus | 1 | ALA4190175 | cell-based format | Scientific Literature | |
| 15. | ALA4190635 | ADME | Stability in dog plasma | Canis lupus familiaris | 1 | ALA4190175 | cell-free format | Scientific Literature | |
| 16. | ALA4190636 | ADME | Stability in rat plasma | Rattus norvegicus | 1 | ALA4190175 | cell-free format | Scientific Literature | |
| 17. | ALA4190637 | Physicochemical | Kinetic solubility of the compound at pH 6.5 | 1 | ALA4190175 | small-molecule physicochemical format | Scientific Literature | ||
| 18. | ALA4190638 | Physicochemical | Thermodynamic solubility of the compound | 1 | ALA4190175 | small-molecule physicochemical format | Scientific Literature | ||
| 19. | ALA4190639 | ADME | Fraction unbound in human plasma | Homo sapiens | 1 | ALA4190175 | cell-free format | Scientific Literature | |
| 20. | ALA4190640 | ADME | Fraction unbound in dog plasma | Canis lupus familiaris | 1 | ALA4190175 | cell-free format | Scientific Literature |
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