| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4187420 | B | Inhibition of N-terminal GST-HIS6 fusion protein tagged human CDK7 (M1 to F346 residues)/N-terminal HIS6-tagged human Cyclin-H (M1 to L323 residues)/N-terminal HIS6-tagged human MAT1 (M1 to S306 residues) expressed in Sf9 cells at 1 uM using RB-CTF substrate and ATP incubated for 1 hr by fluorescent polarization assay | Homo sapiens | 10 | ALA4184207 | cell-based format | Scientific Literature | |
| 2. | ALA4187421 | B | Inhibition of N-terminal GST-HIS6 fusion protein tagged human full length CDK9 (M1 to F372 residues)/N-terminal GST-HIS6 fusion protein tagged human Cyclin-T1 (M1 to K726 residues) expressed in Sf9 cells at 10 uM using TAMRA-Rbtide substrate and ATP incubated for 1 hr by fluorescent polarization assay | Homo sapiens | 53 | ALA4184207 | cell-based format | Scientific Literature | |
| 3. | ALA4187422 | B | Inhibition of human full length CDK2 (M1 to L298 residues)/human full length Cyclin-A2 (M1 to L432 residues) expressed in Sf9 cells at 1 uM using TAMRA-histone H1-derived peptide substrate and ATP incubated for 1 hr by fluorescent polarization assay | Homo sapiens | 10 | ALA4184207 | cell-based format | Scientific Literature | |
| 4. | ALA4187423 | B | Inhibition of human PLK1 kinase domain using 5-TAMRA-RGSFNDTLDFD-NH2 substrate and ATP incubated for 90 mins by fluorescent polarization assay | Homo sapiens | 10 | ALA4184207 | single protein format | Scientific Literature |
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