# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4178003 | B | Inhibition of human PKCalpha (1 to 672 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
2. | ALA4178004 | B | Inhibition of human PAK5 (2 to 719 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
3. | ALA4178005 | B | Inhibition of human PHKgamma1 (2 to 297 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
4. | ALA4178006 | B | Inhibition of recombinant Cryptosporidium parvum FIKK using RRRAPSFYRK peptide as substrate by NADH coupled LDH-PK ATPase assay | Cryptosporidium parvum | 20 | ALA4177526 | assay format | Scientific Literature | |
5. | ALA4178007 | B | Inhibition of Cryptosporidium parvum CDPK1 using PLARTLSVAGLPGKK peptide as substrate by NADH coupled LDH-PK ATPase assay | Cryptosporidium parvum | 20 | ALA4177526 | assay format | Scientific Literature | |
6. | ALA4178037 | B | Selectivity ratio of IC50 for Cryptosporidium parvum CDPK1 to IC50 for recombinant Cryptosporidium parvum FIKK | Cryptosporidium parvum | 1 | ALA4177526 | assay format | Scientific Literature | |
7. | ALA4178038 | B | Inhibition of recombinant Cryptosporidium parvum FIKK assessed as change in melting temperature at 50 uM by differential static light scattering method | Cryptosporidium parvum | 9 | ALA4177526 | assay format | Scientific Literature | |
8. | ALA4178040 | B | Inhibition of MAP4K5 (unknown origin) assessed as residual activity at 500 nM relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
9. | ALA4178041 | B | Inhibition of human S6K1 T412E mutant (1 to 421 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
10. | ALA4178042 | B | Inhibition of human MARK2 (2 to 691 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
11. | ALA4178043 | B | Inhibition of human JNK1 (1 to 384 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
12. | ALA4178044 | B | Inhibition of human GCK (2 to 812 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
13. | ALA4178045 | B | Inhibition of human DYRK1A (1 to 502 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
14. | ALA4178046 | B | Inhibition of human HIPK2 (165 to 564 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
15. | ALA4178047 | B | Inhibition of human RSK1 (1 to 735 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
16. | ALA4178048 | B | Inhibition of human PKBbeta (120 to 481 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
17. | ALA4178049 | B | Inhibition of JAK2 (unknown origin) assessed as residual activity at 500 nM relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
18. | ALA4178050 | B | Inhibition of human TTBK2 (1 to 450 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
19. | ALA4178051 | B | Inhibition of human CAMKKbeta (1 to 541 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature | |
20. | ALA4178052 | B | Inhibition of human SGK1 (60 to 431 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | single protein format | Scientific Literature |