| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4195064 | A | Agonist activity at GAL4 DNA-binding domain-tagged RARalpha (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs by luciferase reporter gene assay | Homo sapiens | 25 | ALA4190387 | cell-based format | Scientific Literature | |
| 2. | ALA4195068 | A | Intrinsic clearance in cryopreserved human hepatocytes assessed per million cells at 1 uM incubated up to 90 mins by LC-MS/MS method | Homo sapiens | 14 | ALA4190387 | cell-based format | Scientific Literature | |
| 3. | ALA4195069 | P | Chromatographic hydrophobicity index, log D of the compound at pH 6.5 by HPLC method | 13 | ALA4190387 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA4195070 | A | Unbound fraction in plasma (unknown origin) | Not specified | 34 | ALA4190387 | cell-free format | Scientific Literature | |
| 5. | ALA4195071 | B | Inverse agonist activity at GAL4 DNA-binding domain-tagged RARgamma (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs by luciferase reporter gene assay | Homo sapiens | 2 | ALA4190387 | cell-based format | Scientific Literature | |
| 6. | ALA4195072 | B | Inverse agonist activity at GAL4 DNA-binding domain-tagged RARabetaa (unknown origin) ligand-binding domain expressed in human HG5LN cells incubated for 18 hrs by luciferase reporter gene assay | Homo sapiens | 2 | ALA4190387 | cell-based format | Scientific Literature |
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