# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4200610 | Binding | Inhibition of human kidney uPA using Z-Gly-Gly-Arg-AMC as substrate measured over 15 mins by fluorescence assay | Homo sapiens | 30 | ALA4196166 | single protein format | Scientific Literature | |
2. | ALA4200611 | Binding | Inhibition of human kidney uPA using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
3. | ALA4200612 | Binding | Inhibition of tPA (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
4. | ALA4200613 | Binding | Inhibition of plasmin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
5. | ALA4200614 | Binding | Inhibition of thrombin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
6. | ALA4200615 | Binding | Inhibition of human plasma kallikrein using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
7. | ALA4200616 | Binding | Inhibition of factor 11a (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
8. | ALA4200617 | Binding | Inhibition of factor 10a (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
9. | ALA4200618 | Binding | Inhibition of trypsin (unknown origin) using chromogenic H-D-Ile-L-Pro-L-Arg-p-nitoraniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | protein format | Scientific Literature | |
10. | ALA4200619 | Binding | Inhibition of activated protein C (unknown origin) using chromogenic L-pyroGlu-L-Pro-L-Arg-p-nitroaniline as substrate by fluorescence assay | Homo sapiens | 4 | ALA4196166 | single protein format | Scientific Literature | |
11. | ALA4200620 | Binding | Inhibition of plasma kallikrein (unknown origin) at 10 nM to 33.3 uM after 30 mins by gel-based ABPP assay | Homo sapiens | 2 | ALA4196166 | single protein format | Scientific Literature | |
12. | ALA4200621 | Binding | Inhibition of trypsin (unknown origin) at 10 nM to 33.3 uM after 30 mins by gel-based ABPP assay | Homo sapiens | 3 | ALA4196166 | protein format | Scientific Literature | |
13. | ALA4200626 | Functional | Cytotoxicity against human MDA-MB-231 cells assessed as reduction in cell viability after 48 hrs by CellTiter 96 Aqueous One solution cell proliferation assay | Homo sapiens | 5 | ALA4196166 | cell-based format | Scientific Literature | |
14. | ALA4200627 | Functional | Cytotoxicity against human HepG2 cells assessed as reduction in cell viability after 48 hrs by CellTiter 96 Aqueous One solution cell proliferation assay | Homo sapiens | 5 | ALA4196166 | cell-based format | Scientific Literature | |
15. | ALA4200628 | ADME | Cytotoxicity against HEK293 cells assessed as reduction in cell viability after 48 hrs by CellTiter 96 Aqueous One solution cell proliferation assay | Homo sapiens | 5 | ALA4196166 | cell-based format | Scientific Literature | |
16. | ALA4200629 | Functional | Cytotoxicity against human HT1080 cells assessed as reduction in cell viability after 48 hrs by CellTiter 96 Aqueous One solution cell proliferation assay | Homo sapiens | 5 | ALA4196166 | cell-based format | Scientific Literature | |
17. | ALA4200630 | Physicochemical | Lipophilicity, log D of the compound at pH 7.4 | 4 | ALA4196166 | small-molecule physicochemical format | Scientific Literature | ||
18. | ALA4200632 | Binding | Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assay | Mus musculus | 4 | ALA4196166 | single protein format | Scientific Literature | |
19. | ALA4200633 | Binding | Selectivity ratio of IC50 for mouse uPA to Ki for human uPA | 4 | ALA4196166 | assay format | Scientific Literature | ||
20. | ALA4200634 | ADME | Inhibition of S-3969-stimulated recombinant human ENaC alpha subunit expressed in HEK293 cells at 10 uM preincubated for 5 mins followed by S-3969 stimulation by FLIPR assay | Homo sapiens | 6 | ALA4196166 | cell-based format | Scientific Literature |
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