# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4185001 | Binding | Inhibition of 20s constitutive proteasome beta1 caspase-like activity in human erythrocytes using Z-Leu-Leu-Glu-AMC as substrate after 10 mins by fluorescence assay | Homo sapiens | 2 | ALA4184119 | cell-based format | Scientific Literature | |
2. | ALA4185002 | Binding | Inhibition of 20s constitutive proteasome beta2 trypsin-like activity in human erythrocytes using Boc-Leu-Arg-Arg-AMC as substrate at 50 uM after 10 mins by fluorescence assay relative to control | Homo sapiens | 10 | ALA4184119 | cell-based format | Scientific Literature | |
3. | ALA4185005 | Binding | Inhibition of 20s immunoproteasome beta2 trypsin-like activity in human spleen using Boc-Leu-Arg-Arg-AMC as substrate after 10 mins by fluorescence assay | Homo sapiens | 4 | ALA4184119 | single protein format | Scientific Literature | |
4. | ALA4185006 | Binding | Inhibition of 20s constitutive proteasome beta5 chymotrypsin-like activity in human erythrocytes using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM after 10 mins by fluorescence assay relative to control | Homo sapiens | 8 | ALA4184119 | cell-based format | Scientific Literature | |
5. | ALA4185008 | Binding | Inhibition of 20s immunoproteasome beta5 chymotrypsin-like activity in human spleen using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM after 10 mins by fluorescence assay relative to control | Homo sapiens | 6 | ALA4184119 | single protein format | Scientific Literature | |
6. | ALA4185010 | Binding | Inhibition of 20s immunoproteasome beta1 caspase-like activity in human spleen using Ac-Pro-Ala-Leu-AMC as substrate at 50 uM after 10 mins by fluorescence assay relative to control | Homo sapiens | 9 | ALA4184119 | single protein format | Scientific Literature |