| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4201797 | B | Inhibition of human recombinant MMP1 catalytic domain at 100 uM using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 2. | ALA4201799 | B | Slow binding inhibition of human recombinant MMP2 using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 3. | ALA4201800 | B | Inhibition of human recombinant MMP3 catalytic domain at 100 uM using MOCAc-Arg-Pro-Lys-Pro-Val-Glu-Nva-Trp-Arg-Lys(Dnp)-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 4. | ALA4201801 | B | Inhibition of human recombinant MMP7 at 100 uM using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 5. | ALA4201802 | B | Non-competitive inhibition of human recombinant MMP8 catalytic domain using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 6. | ALA4201803 | B | Slow binding inhibition of human recombinant MMP9 catalytic domain using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 7. | ALA4201804 | B | Slow binding inhibition of human recombinant MMP14 catalytic domain using MOCAc-Pro-Leu-Gly-Leu-A2pr(Dnp)-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 8. | ALA4201805 | B | Inhibition of human recombinant ADAM9 at 100 uM using Mca-Pro-Leu-Ala-Gln-Ala-Val-Dpa-Arg-Ser-Ser-Ser-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 9. | ALA4201806 | B | Inhibition of human recombinant ADAM10 at 100 uM using Mca-Lys-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 substrate | Homo sapiens | 3 | ALA4196209 | single protein format | Scientific Literature | |
| 10. | ALA4201807 | B | Selectivity index, ratio of Ki for non-competitive inhibition of human recombinant MMP8 catalytic domain to KI for slow binding inhibition of human recombinant MMP9 catalytic domain | Homo sapiens | 3 | ALA4196209 | assay format | Scientific Literature | |
| 11. | ALA4201812 | F | Induction of wound healing in db/db BKS.Cg-Dock7m+/+ Lepr db/J mouse model of full-thickness excision at 50 ug/wound/day for 14 days dosed topically 1 day after wound creation | Mus musculus | 3 | ALA4196209 | organism-based format | Scientific Literature | |
| 12. | ALA4201813 | F | Induction of wound healing in db/db BKS.Cg-Dock7m+/+ Lepr db/J mouse model of full-thickness excision assessed as increase in re-epithelialization at 50 ug/wound/day for 14 days dosed topically 1 day after wound creation by H and E staining | Mus musculus | 3 | ALA4196209 | organism-based format | Scientific Literature | |
| 13. | ALA4201814 | F | Inhibition of MMP9 activity in db/db BKS.Cg-Dock7m+/+ Lepr db/J mouse model of full-thickness excision using DQ-gelatin substrate at 50 ug/wound/day for 14 days dosed topically 1 day after wound creation by in-situ zymography | Mus musculus | 3 | ALA4196209 | organism-based format | Scientific Literature | |
| 14. | ALA4201815 | F | Inhibition of MMP8 activity in db/db BKS.Cg-Dock7m+/+ Lepr db/J mouse model of full-thickness excision using DQ-collagen substrate at 50 ug/wound/day for 14 days dosed topically 1 day after wound creation by in-situ zymography | Mus musculus | 3 | ALA4196209 | organism-based format | Scientific Literature |
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