| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4192331 | B | Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 2. | ALA4192332 | B | Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting method | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 3. | ALA4192334 | F | Cytoprotection against H2O2-induced oxidative damage in differentiated human IMR32 cells at 0.1 to 1 uM preincubated for 24 hrs followed by H2O2 addition measured after 1 hr by DCF-DA staining based fluorescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA4192343 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Vmax at 3 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 19490 +/- 852 cpm) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA4192344 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Vmax at 6 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 19490 +/- 852 cpm) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4192345 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Vmax at 9 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 19490 +/- 852 cpm) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA4192346 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Vmax at 12 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 19490 +/- 852 cpm) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4192347 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Km at 3 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 9.9 +/- 0.9 uM) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4192348 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Km at 6 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 9.9 +/- 0.9 uM) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4192349 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Km at 9 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 9.9 +/- 0.9 uM) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4192350 | B | Inhibition of recombinant human His-tagged GSK3beta assessed as substrate Km at 12 uM using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method (Rvb = 9.9 +/- 0.9 uM) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4192351 | B | Non-competitive inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 13. | ALA4192352 | A | Cytotoxicity against human IMR32 cells assessed as reduction in cell viability at 0.1 to 50 uM after 24 hrs by LDH release assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 14. | ALA4192354 | A | Cytotoxicity against human IMR32 cells assessed as effect on cellular morphology at 0.1 to 50 uM after 24 hrs | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA4192355 | F | Cytoprotection against H2O2-induced oxidative damage in human IMR32 cells at 0.1 to 1 uM preincubated for 24 hrs followed by H2O2 addition measured after 1 hr by DCF-DA staining based fluorescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature |
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