# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4195968 | Functional | Agonist activity at SSTR1 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced CRE promoter activity at 10 to 1000 nM by luciferase reporter gene assay | Homo sapiens | 3 | ALA4190409 | cell-based format | Scientific Literature | |
2. | ALA4195969 | Functional | Agonist activity at SSTR2 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced CRE promoter activity at 10 to 1000 nM by luciferase reporter gene assay | Homo sapiens | 4 | ALA4190409 | cell-based format | Scientific Literature | |
3. | ALA4195970 | Functional | Agonist activity at SSTR3 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced CRE promoter activity at 10 to 1000 nM by luciferase reporter gene assay | Homo sapiens | 4 | ALA4190409 | cell-based format | Scientific Literature | |
4. | ALA4195971 | Functional | Agonist activity at SSTR4 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced CRE promoter activity at 10 to 1000 nM by luciferase reporter gene assay | Homo sapiens | 3 | ALA4190409 | cell-based format | Scientific Literature | |
5. | ALA4195972 | Functional | Agonist activity at SSTR5 (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced CRE promoter activity at 10 to 1000 nM by luciferase reporter gene assay | Homo sapiens | 4 | ALA4190409 | cell-based format | Scientific Literature | |
6. | ALA4195973 | ADME | Drug uptake in HEK293 cells co-expressing SSTR1 (unknown origin) and RFP assessed as SSTR1-mediated drug accumulation by measuring mean fluorescence intensity measured after 30 mins by fluorescence microscopic analysis (Rvb = 1.1 No_unit) | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
7. | ALA4195974 | ADME | Drug uptake in HEK293 cells co-expressing SSTR2 (unknown origin) and RFP assessed as SSTR2-mediated drug accumulation by measuring mean fluorescence intensity measured after 30 mins by fluorescence microscopic analysis (Rvb = 1.1 No_unit) | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
8. | ALA4195975 | ADME | Drug uptake in HEK293 cells co-expressing SSTR3 (unknown origin) and RFP assessed as SSTR3-mediated drug accumulation by measuring mean fluorescence intensity measured after 30 mins by fluorescence microscopic analysis (Rvb = 1.1 No_unit) | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
9. | ALA4195976 | ADME | Drug uptake in HEK293 cells co-expressing SSTR4 (unknown origin) and RFP assessed as SSTR4-mediated drug accumulation by measuring mean fluorescence intensity measured after 30 mins by fluorescence microscopic analysis (Rvb = 1.1 No_unit) | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
10. | ALA4195977 | ADME | Drug uptake in HEK293 cells co-expressing SSTR5 (unknown origin) and RFP assessed as SSTR5-mediated drug accumulation by measuring mean fluorescence intensity measured after 30 mins by fluorescence microscopic analysis (Rvb = 1.1 No_unit) | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
11. | ALA4195978 | ADME | Drug uptake in HEK293 cells co-expressing SSTR2 (unknown origin) and RFP assessed as SSTR2-mediated drug accumulation by measuring mean fluorescence intensity at 400 nM measured after 15 mins in presence of SSTR2 agonist octreotide by fluorescence assay | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
12. | ALA4195979 | ADME | Drug uptake in HEK293 cells co-expressing SSTR4 (unknown origin) and RFP assessed as SSTR4-mediated drug accumulation by measuring mean fluorescence intensity at 400 nM measured after 15 mins in presence of SSTR2 agonist octreotide by fluorescence assay | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
13. | ALA4195981 | ADME | Drug uptake in human PANC1 cells assessed as SSTR2/SSTR5-mediated drug accumulation measured up to 24 hrs by DAPI staining based confocal microscopic analysis | Homo sapiens | 1 | ALA4190409 | cell-based format | Scientific Literature | |
14. | ALA4195982 | ADME | Drug uptake in human Capan1 cells assessed as SSTR2/SSTR5-mediated drug accumulation measured up to 24 hrs by DAPI staining based confocal microscopic analysis | Homo sapiens | 2 | ALA4190409 | cell-based format | Scientific Literature |