Inhibition of N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain expressed in Baculovirus infected Sf9 insect cells using FAM-cGMP as substrate after 1 hr by fluorescence polarization assay
Selectivity ratio of IC50 for N-terminal GST-tagged full length recombinant human PDE1A to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain
Selectivity ratio of IC50 for N-terminal FLAG-tagged human PDE2A1 (2 to 941 residues) to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain
Selectivity ratio of IC50 for N-terminal GST-tagged recombinant human PDE3B (592 end residues) to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain
Selectivity ratio of IC50 for N-terminal GST-tagged full length recombinant human PDE4A1A to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain
Selectivity ratio of IC50 for N-terminal GST-tagged full length recombinant human PDE6C to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain
Selectivity ratio of IC50 for N-terminal GST-tagged full length recombinant human PDE11A to IC50 for N-terminal GST-tagged full length recombinant human PDE5A1 catalytic domain