#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4178741	Functional	Antagonist activity at human GPR4 expressed in human HeLa cells assessed as inhibition of IBMX-induced cAMP accumulation after 15 mins by HTRF assay	Homo sapiens	13	ALA4177561	cell-based format	Scientific Literature
2.	ALA4178742	Binding	Displacement of [3H]dofetilide from recombinant human ERG expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting method	Homo sapiens	13	ALA4177561	cell-based format	Scientific Literature
3.	ALA4178743	Binding	Selectivity ratio of IC50 for displacement of [3H]dofetilide from recombinant human ERG expressed in HEK293 cell membranes to IC50 for human GPR4 expressed in HeLa cells	Homo sapiens	13	ALA4177561	cell-based format	Scientific Literature
4.	ALA4178744	Binding	Displacement of [3H]-R(-)-alpha-Methyl[imidazole-2.5(n)]histamine from human recombinant histamine H3 receptor expressed in CHOK1 cell membranes after 1 hr by scintillation counting method	Homo sapiens	13	ALA4177561	cell-based format	Scientific Literature
5.	ALA4178745	ADME	Clearance in Sprague-Dawley rat at 1 mg/kg, iv	Rattus norvegicus	11	ALA4177561	organism-based format	Scientific Literature
6.	ALA4178746	ADME	Dose normalized AUC in Sprague-Dawley rat at 3 mg/kg, po	Rattus norvegicus	11	ALA4177561	organism-based format	Scientific Literature
7.	ALA4178747	Functional	Antagonist activity at rat GPR4 expressed in HEK cells assessed as inhibition of IBMX-induced cAMP accumulation after 15 mins by HTRF assay	Rattus norvegicus	3	ALA4177561	cell-based format	Scientific Literature
8.	ALA4178748	Functional	Antiarthritic activity in Lewis rat antigen-induced arthritis model assessed as inhibition of arthritic knee swelling at 30 mg/kg, po bid for 7 days dosed after 21 and 14 days of methylated BSA and complete Freund's adjuvant sensitization measured after 7 days post dose relative to 1 mg/kg, po qd dexamethasone	Rattus norvegicus	3	ALA4177561	organism-based format	Scientific Literature
9.	ALA4178757	Functional	Antagonist activity at human GPR4 expressed in human HeLa cells assessed as inhibition of IBMX-induced cAMP accumulation after 15 mins in presence of 40% rat plasma by HTRF assay	Homo sapiens	3	ALA4177561	cell-based format	Scientific Literature
10.	ALA4178758	Binding	Ratio of IC50 for human GPR4 expressed in human HeLa cells in presence of 40% rat plasma to IC50 for human GPR4 expressed in human HeLa in absence of 40% rat plasma	Homo sapiens	3	ALA4177561	cell-based format	Scientific Literature
11.	ALA4178760	ADME	Protein binding in rat plasma	Rattus norvegicus	2	ALA4177561	cell-free format	Scientific Literature
12.	ALA4178761	ADME	Protein binding in human plasma	Homo sapiens	2	ALA4177561	cell-free format	Scientific Literature