| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4193339 | B | Displacement of 7-methoxy-[3H]-prazosin from human alpha1D-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintillation counting method | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
| 2. | ALA4193340 | B | Displacement of 7-methoxy-[3H]-prazosin from human alpha1B-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintillation counting method | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 3. | ALA4193341 | B | Displacement of 7-methoxy-[3H]-prazosin from human alpha1A-adrenoreceptor expressed in CHOK1 cell membranes after 60 mins by TopCount liquid scintillation counting method | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 4. | ALA4193342 | B | Selectivity ratio of Ki for human alpha1A-adrenoreceptor to Ki for human alpha1D-adrenoreceptor | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 5. | ALA4193343 | B | Selectivity ratio of Ki for human alpha1B-adrenoreceptor to Ki for human alpha1D-adrenoreceptor | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 6. | ALA4193344 | F | Antagonist activity at alpha1D-adrenoreceptor in Wistar rat bladder strips assessed as relaxation of PHE-induced contractile response after 30 mins | Rattus norvegicus | 6 | assay format | Scientific Literature | ||
| 7. | ALA4193345 | A | Intrinsic clearance in human liver microsomes at 10 uM after 15 to 30 mins by LC-MS/MS analysis | Homo sapiens | 13 | microsome format | Scientific Literature | ||
| 8. | ALA4193346 | A | Inhibition of human microsomal CYP3A4 at 10 uM after 10 mins by LC-MS/MS analysis relative to control | Homo sapiens | 13 | assay format | Scientific Literature |
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