| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4220820 | B | Inhibition of recombinant human JAK1 (866-end residues) in presence of ATP | Homo sapiens | 38 | ALA4219073 | single protein format | Scientific Literature | |
| 2. | ALA4220821 | A | Inhibition of recombinant human JAK2 (808-end residues) in presence of ATP | Homo sapiens | 38 | ALA4219073 | single protein format | Scientific Literature | |
| 3. | ALA4220822 | B | Selectivity index, ratio of IC50 for recombinant human JAK2 (808-end residues) to IC50 for recombinant human JAK1 (866-end residues) | Homo sapiens | 38 | ALA4219073 | assay format | Scientific Literature | |
| 4. | ALA4220823 | B | Inhibition of human ERG expressed in HEK293 cells by automated patch clamp method | Homo sapiens | 2 | ALA4219073 | cell-based format | Scientific Literature | |
| 5. | ALA4220824 | A | Metabolic stability in human liver microsomes assessed as parent compound remaining after 30 mins | Homo sapiens | 4 | ALA4219073 | microsome format | Scientific Literature | |
| 6. | ALA4220825 | A | Metabolic stability in dog liver microsomes assessed as parent compound remaining after 30 mins | Canis lupus familiaris | 4 | ALA4219073 | microsome format | Scientific Literature | |
| 7. | ALA4220826 | A | Metabolic stability in rat liver microsomes assessed as parent compound remaining after 30 mins | Rattus norvegicus | 4 | ALA4219073 | microsome format | Scientific Literature | |
| 8. | ALA4220827 | A | Metabolic stability in mouse liver microsomes assessed as parent compound remaining after 30 mins | Mus musculus | 4 | ALA4219073 | microsome format | Scientific Literature | |
| 9. | ALA4220828 | A | Protein binding in human plasma | Homo sapiens | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 10. | ALA4220829 | A | Protein binding in rat plasma | Rattus norvegicus | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 11. | ALA4220830 | A | Metabolic stability in human plasma assessed as parent compound remaining after 30 mins | Homo sapiens | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 12. | ALA4220831 | A | Metabolic stability in human plasma assessed as parent compound remaining after 120 mins | Homo sapiens | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 13. | ALA4220832 | A | Metabolic stability in rat plasma assessed as parent compound remaining after 120 mins | Rattus norvegicus | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 14. | ALA4220833 | A | Metabolic stability in rat plasma assessed as parent compound remaining after 30 mins | Rattus norvegicus | 1 | ALA4219073 | cell-free format | Scientific Literature | |
| 15. | ALA4220834 | A | Apparent permeability from apical to basolateral side in human Caco2 cells | Homo sapiens | 1 | ALA4219073 | cell-based format | Scientific Literature | |
| 16. | ALA4220835 | A | Apparent permeability from basolateral to apical side in human Caco2 cells | Homo sapiens | 1 | ALA4219073 | cell-based format | Scientific Literature | |
| 17. | ALA4220836 | A | Efflux ratio of apparent permeability in human Caco2 cells | Homo sapiens | 1 | ALA4219073 | cell-based format | Scientific Literature | |
| 18. | ALA4220837 | A | Inhibition of CYP1A2 (unknown origin) assessed as residual activity at 10 uM relative to control | Homo sapiens | 1 | ALA4219073 | single protein format | Scientific Literature | |
| 19. | ALA4220838 | A | Inhibition of CYP2C9 (unknown origin) assessed as residual activity at 10 uM relative to control | Homo sapiens | 1 | ALA4219073 | single protein format | Scientific Literature | |
| 20. | ALA4220839 | A | Inhibition of CYP2C19 (unknown origin) assessed as residual activity at 10 uM relative to control | Homo sapiens | 1 | ALA4219073 | single protein format | Scientific Literature |
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