| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4221488 | B | Inhibition of adenosine receptor (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4219104 | protein format | Scientific Literature | |
| 2. | ALA4221489 | B | Inhibition of recombinant human GlyT1 expressed in CHO cells assessed as reduction in [3H]glycine uptake pretreated for 15 mins followed by [3H]glycine addition measured after 2 hrs by Topcount method | Homo sapiens | 45 | ALA4219104 | cell-based format | Scientific Literature | |
| 3. | ALA4221490 | P | Equilibrium solubility of the compound in phosphate buffer at pH 7.4 by UV-HPLC analysis | 16 | ALA4219104 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA4221491 | P | Octanol-water partition coefficient, log D of the compound at pH 7.4 | 38 | ALA4219104 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4221492 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 39 | ALA4219104 | microsome format | Scientific Literature | |
| 6. | ALA4221493 | A | Efflux ratio of permeability in MDCK cells expressing P-gp | Canis lupus familiaris | 25 | ALA4219104 | cell-based format | Scientific Literature | |
| 7. | ALA4221494 | A | Intrinsic clearance in Sprague-Dawley rat liver microsomes | Rattus norvegicus | 1 | ALA4219104 | microsome format | Scientific Literature | |
| 8. | ALA4221495 | A | Protein binding in Sprague-Dawley rat plasma assessed as unbound fraction by equilibrium dialysis method | Rattus norvegicus | 1 | ALA4219104 | cell-free format | Scientific Literature | |
| 9. | ALA4221496 | A | Clearance in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 10. | ALA4221497 | A | Volume of distribution at steady state in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 11. | ALA4221498 | A | Half life in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 12. | ALA4221499 | A | Ratio of drug level in brain to plasma in Sprague-Dawley rat at 3 umol/kg, iv | Rattus norvegicus | 1 | ALA4219104 | cell-free format | Scientific Literature | |
| 13. | ALA4221500 | A | Cmax in Sprague-Dawley rat at 9 umol/kg, po | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 14. | ALA4221501 | A | Tmax in Sprague-Dawley rat at 9 umol/kg, po | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 15. | ALA4221502 | A | Oral bioavailability in Sprague-Dawley rat at 9 umol/kg | Rattus norvegicus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 16. | ALA4221503 | A | Ratio of drug level in brain to plasma in sc dosed CD-1 mouse | Mus musculus | 1 | ALA4219104 | organism-based format | Scientific Literature | |
| 17. | ALA4221504 | A | Protein binding in CD-1 mouse plasma assessed as unbound fraction | Mus musculus | 1 | ALA4219104 | cell-free format | Scientific Literature | |
| 18. | ALA4221505 | B | Inhibition of DAT transporter (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4219104 | single protein format | Scientific Literature | |
| 19. | ALA4221506 | B | Inhibition of NET transporter (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4219104 | single protein format | Scientific Literature | |
| 20. | ALA4221507 | B | Inhibition of SERT transporter (unknown origin) at 10 uM | Homo sapiens | 1 | ALA4219104 | single protein format | Scientific Literature |
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