# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4236637 | B | Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
2. | ALA4236638 | B | Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
3. | ALA4236639 | B | Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
4. | ALA4236640 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
5. | ALA4236641 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM after 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
6. | ALA4236645 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM for 4 hrs at pH 5 to 9 at room temperature by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
7. | ALA4236646 | B | Irreversible inhibition of N-terminal His-tagged BRD4 (BD1)(unknown origin) assessed as change in mass by measuring unbound protein mass by MALDI-TOF mass spectrometric analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA4236665 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature incubated for 4 hrs in presence of increasing concentrations of cysteine amino acids by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
9. | ALA4236666 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature incubated for 4 hrs in presence of increasing concentrations of methionine by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
10. | ALA4236667 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM incubated for 4 h followed by 3 freeze-thaw cycles by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
11. | ALA4236668 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM incubated for 4 hrs at 37 degC by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
12. | ALA4236669 | B | Binding affinity to N-terminal His-tagged BRD4 (BD1) (unknown origin) assessed as change in melting temperature at 100 uM incubated for 4 hrs at room tempaerature by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA4236671 | B | Binding affinity to PHIP (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
14. | ALA4236672 | B | Binding affinity to BRG1 (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
15. | ALA4236673 | B | Binding affinity to TAF1(2) (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
16. | ALA4236674 | B | Binding affinity to P300 (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
17. | ALA4236675 | B | Binding affinity to BRPF1 (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
18. | ALA4236676 | B | Binding affinity to CREBBP (unknown origin) assessed as change in melting temperature at 100 uM after 0.5 to 4 hrs by SYPRO orange protein staining-based thermal denaturation assay | Homo sapiens | 4 | single protein format | Scientific Literature |