# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4236727 | B | Inhibition of recombinant human PACE4 expressed in S2 insect cells using pyroGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate after 1 hr by spectrofluorometry | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
2. | ALA4236732 | A | Cytotoxicity against human DU145 cells assessed as effect on live cells up to 100 uM after 1.5 hrs by propidium iodide-staining based FACS analysis | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
3. | ALA4236735 | F | Antiproliferative activity against human LNCAP cells up to 300 uM after 72 hrs by MTT assay relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
4. | ALA4236736 | F | Antiproliferative activity against human DU145 cells after 72 hrs by MTT assay | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
5. | ALA4236738 | B | Selectivity ratio of Ki for recombinant human furin to Ki for recombinant human PACE4 | Homo sapiens | 27 | assay format | Scientific Literature | ||
6. | ALA4236739 | B | Inhibition of recombinant human furin expressed in S2 insect cells using pyroGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate after 1 hr by spectrofluorometry | Homo sapiens | 27 | cell-based format | Scientific Literature |