| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4268221 | B | Inhibition of human JAK2 using poly(Glu:Tyr)(4:1) as substrate preincubated for 20 mins followed by [gamma33P]ATP addition measured after 120 mins by ion exchange filter paper method | Homo sapiens | 29 | single protein format | Scientific Literature | ||
| 2. | ALA4268222 | B | Inhibition of HDAC1 (unknown origin) using Arg-His-Lys-Lys(Ac) as substrate preincubated with enzyme followed by substrate addition for 2 hrs and measured for 1.5 hrs at 15 mins time interval by fluorescence assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 3. | ALA4268223 | B | Inhibition of HDAC6 (unknown origin) using Arg-His-Lys-Lys(Ac) as substrate preincubated with enzyme followed by substrate addition for 2 hrs and measured for 1.5 hrs at 15 mins time interval by fluorescence assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 4. | ALA4268237 | A | Antiproliferative activity against human AC10 cells after 72 hrs by MTT assay | Homo sapiens | 20 | cell-based format | Scientific Literature | ||
| 5. | ALA4268238 | A | Antiproliferative activity against mouse TAMH cells after 72 hrs by MTT assay | Mus musculus | 20 | cell-based format | Scientific Literature | ||
| 6. | ALA4268239 | T | Selectivity index, ratio of CC50 for human AC10 cells to IC50 for human HCT116 cells | Homo sapiens | 18 | assay format | Scientific Literature | ||
| 7. | ALA4268240 | T | Selectivity index, ratio of CC50 for mouse TAMH cells to IC50 for human HCT116 cells | 18 | assay format | Scientific Literature | |||
| 8. | ALA4268241 | T | Selectivity index, ratio of CC50 for human AC10 cells to IC50 for human MDA-MB-231 cells | Homo sapiens | 19 | assay format | Scientific Literature | ||
| 9. | ALA4268242 | T | Selectivity index, ratio of CC50 for mouse TAMH cells to IC50 for human MDA-MB-231 cells | 19 | assay format | Scientific Literature | |||
| 10. | ALA4268243 | T | Selectivity index, ratio of CC50 for human AC10 cells to IC50 for human MCF7 cells | Homo sapiens | 19 | assay format | Scientific Literature | ||
| 11. | ALA4268244 | T | Selectivity index, ratio of CC50 for mouse TAMH cells to IC50 for human MCF7 cells | 19 | assay format | Scientific Literature | |||
| 12. | ALA4268245 | T | Selectivity index, ratio of CC50 for human AC10 cells to IC50 for human PC3 cells | Homo sapiens | 19 | assay format | Scientific Literature | ||
| 13. | ALA4268246 | T | Selectivity index, ratio of CC50 for mouse TAMH cells to IC50 for human PC3 cells | 19 | assay format | Scientific Literature |
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