| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4256413 | B | Irreversible inhibition of human leukocyte elastase assessed as ratio of Kinact to Ki using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 2. | ALA4256414 | B | Inhibition of porcine pancreatic elastase assessed as ratio of Kinact to Ki using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated over 60 mins by spectrophotometric method | Sus scrofa | 2 | protein format | Scientific Literature | ||
| 3. | ALA4256415 | B | Inhibition of bovine chymotrypsin assessed as ratio of Kinact to Ki using Suc-Ala-Ala-Pro-Phe-pNA as substrate incubated over 60 mins by spectrophotometric method | Bos taurus | 1 | assay format | Scientific Literature | ||
| 4. | ALA4256416 | B | Inhibition of bovine factor 10a assessed as product formation at 1 uM using Boc-Ile-Glu-Gly-Arg-AMC as substrate incubated over 60 mins by fluorimetric method | Bos taurus | 3 | single protein format | Scientific Literature | ||
| 5. | ALA4256417 | B | Inhibition of human thrombin assessed as product formation at 1 uM using Z-Gly-Gly-Arg-AMC as substrate incubated over 60 mins by fluorimetric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA4256418 | B | Inhibition of bovine trypsin assessed as product formation at 1 uM using Suc-Ala-Ala-Pro-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Bos taurus | 3 | assay format | Scientific Literature | ||
| 7. | ALA4256419 | B | Inhibition of human cathepsin B assessed as product formation at 1 uM using Z-Arg-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA4256420 | B | Inhibition of human cathepsin L assessed as product formation at 1 uM using Z-Phe-Arg-pNA as substrate incubated over 60 mins by spectrophotometric method | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA4256427 | B | Irreversible inhibition of human leukocyte elastase at 50 nM using MeO-Suc-Ala-Ala-Pro-Val-pNA as substrate incubated for 30 mins followed by substrate addition | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4256428 | B | Binding affinity to human leukocyte elastase at 2.5 uM after 20 mins by in gel fluorescence detection based SDS-PAGE analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4256429 | B | Binding affinity to human leukocyte elastase at 160 ng after 20 mins by in gel fluorescence detection based SDS-PAGE analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4256430 | B | Binding affinity to human leukocyte elastase at 2.5 uM after 20 mins by Coomassie brilliant blue G-250 staining based assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4256431 | B | Binding affinity to human leukocyte elastase at 2.5 uM incubated for 20 mins followed by HEK cell lysate addition by in gel fluorescence detection based SDS-PAGE analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4256432 | B | Binding affinity to human leukocyte elastase at 2.5 uM incubated for 20 mins post HEK cell lysate addition by in gel fluorescence detection based SDS-PAGE analysis | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4256433 | B | Binding affinity to human leukocyte elastase at 2.5 uM incubated for 20 mins followed by HEK cell lysate addition by Coomassie brilliant blue G-250 staining based assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4256434 | B | Binding affinity to human leukocyte elastase at 2.5 uM incubated for 20 mins post HEK cell lysate addition by Coomassie brilliant blue G-250 staining based assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4256435 | B | Inhibition of human leukocyte elastase at 2.5 uM preincubated with sivelestat for 5 mins followed by compound addition measured after 20 mins in presence of sivelestat by in gel fluorescence detection based SDS-PAGE analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4256436 | B | Inhibition of human leukocyte elastase at 2.5 uM preincubated with sivelestat for 5 mins followed by compound addition measured after 20 mins in presence of sivelestat by Coomassie brilliant blue G-250 staining based assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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