| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4266687 | Binding | Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cell membranes after 60 mins by TopCount microplate scintillation counting method | Homo sapiens | 26 | ALA4265879 | cell-based format | Scientific Literature | |
| 2. | ALA4266688 | Binding | Selectivity index, ratio of Ki for human vasopressin V1a receptor to Ki for human vasopressin V1b receptor | Homo sapiens | 16 | ALA4265879 | assay format | Scientific Literature | |
| 3. | ALA4266689 | Binding | Selectivity index, ratio of Ki for human oxytocin receptor to Ki for human vasopressin V1b receptor | Homo sapiens | 16 | ALA4265879 | assay format | Scientific Literature | |
| 4. | ALA4266690 | ADME | Intrinsic clearance in human liver microsomes | Homo sapiens | 23 | ALA4265879 | microsome format | Scientific Literature | |
| 5. | ALA4266691 | ADME | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 23 | ALA4265879 | microsome format | Scientific Literature | |
| 6. | ALA4266692 | ADME | Elimination half life in rat at 2 mg/kg, iv | Rattus norvegicus | 4 | ALA4265879 | organism-based format | Scientific Literature | |
| 7. | ALA4266693 | ADME | Volume of distribution at steady state in rat at 2 mg/kg, iv | Rattus norvegicus | 4 | ALA4265879 | organism-based format | Scientific Literature | |
| 8. | ALA4266694 | ADME | Clearance in rat plasma at 2 mg/kg, iv | Rattus norvegicus | 4 | ALA4265879 | organism-based format | Scientific Literature | |
| 9. | ALA4266695 | ADME | Oral bioavailability in rat at 10 mg/kg | Rattus norvegicus | 3 | ALA4265879 | organism-based format | Scientific Literature | |
| 10. | ALA4266697 | ADME | Ratio of AUC in rat brain to plasma at 10 mg/kg, ip measured after 8 hrs | Rattus norvegicus | 4 | ALA4265879 | organism-based format | Scientific Literature |
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