| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4270237 | A | Drug uptake in C57BL/6N mouse whole blood at 3 mg/kg, po measured at 3 hrs | Mus musculus | 1 | ALA4266056 | organism-based format | Scientific Literature | |
| 2. | ALA4270238 | B | Displacement of (3-125I-Tyr11)-SRIF-28 from human SSTR5 expressed in CHO-K1 cell membranes by filtration binding assay | Homo sapiens | 10 | ALA4266056 | cell-based format | Scientific Literature | |
| 3. | ALA4270239 | B | Displacement of (3-125I-Tyr11)-SRIF-28 from mouse SSTR5 expressed in CHO-K1 cell membranes by filtration binding assay | Mus musculus | 10 | ALA4266056 | cell-based format | Scientific Literature | |
| 4. | ALA4270240 | F | Antagonist activity at human SSTR5 expressed in CHO-K1 cell membranes assessed as reduction in SST-28-induced inhibition of forskolin-stimulated cAMP accumulation by LANCE assay | Homo sapiens | 10 | ALA4266056 | cell-based format | Scientific Literature | |
| 5. | ALA4270241 | F | Antagonist activity at mouse SSTR5 expressed in CHO-K1 cell membranes assessed as reduction in SST-28-induced inhibition of forskolin-stimulated cAMP accumulation by LANCE assay | Mus musculus | 10 | ALA4266056 | cell-based format | Scientific Literature | |
| 6. | ALA4270242 | B | Inhibition of MK-499 binding to human ERG | Homo sapiens | 10 | ALA4266056 | single protein format | Scientific Literature | |
| 7. | ALA4270245 | F | Antidiabetic activity in HFD fed C57BL/6N mouse assessed as decrease in blood glucose AUC at 3 mg/kg administered as single oral dose pretreated for 60 mins followed by glucose challenge measured after 120 mins by OGTT | Mus musculus | 1 | ALA4266056 | organism-based format | Scientific Literature | |
| 8. | ALA4270249 | F | Antagonist activity at human SSTR1 expressed in CHO-K1 cell membranes | Homo sapiens | 3 | ALA4266056 | cell-based format | Scientific Literature | |
| 9. | ALA4270250 | F | Antagonist activity at human SSTR3 expressed in CHO-K1 cell membranes | Homo sapiens | 2 | ALA4266056 | cell-based format | Scientific Literature | |
| 10. | ALA4270251 | F | Antagonist activity at human SSTR2 expressed in CHO-K1 cell membranes | Homo sapiens | 1 | ALA4266056 | cell-based format | Scientific Literature | |
| 11. | ALA4270252 | F | Antagonist activity at human SSTR4 expressed in CHO-K1 cell membranes | Homo sapiens | 1 | ALA4266056 | cell-based format | Scientific Literature | |
| 12. | ALA4270253 | F | Agonist activity at human SSTR5 expressed in CHO-K1 cell membranes assessed as forskolin-stimulated cAMP accumulation at 8.3 uM preincubated for 15 mins followed by forskolin addition measured after 1 hr by LANCE assay | Homo sapiens | 1 | ALA4266056 | cell-based format | Scientific Literature | |
| 13. | ALA4270254 | B | Inhibition of IKs (unknown origin) | Homo sapiens | 1 | ALA4266056 | single protein format | Scientific Literature | |
| 14. | ALA4270255 | B | Inhibition of Cav1.2 (unknown origin) | Homo sapiens | 1 | ALA4266056 | single protein format | Scientific Literature | |
| 15. | ALA4270256 | B | Inhibition of Nav1.5 (unknown origin) | Homo sapiens | 1 | ALA4266056 | single protein format | Scientific Literature | |
| 16. | ALA4270257 | B | Inhibition of prostanoid DP receptor (unknown origin) | Homo sapiens | 1 | ALA4266056 | single protein format | Scientific Literature | |
| 17. | ALA4270258 | A | Fraction unbound in rat plasma at 0.1 uM using [3H]-labeled compound | Rattus norvegicus | 1 | ALA4266056 | cell-free format | Scientific Literature | |
| 18. | ALA4270259 | A | Fraction unbound in dog plasma at 0.1 uM using [3H]-labeled compound | Canis lupus familiaris | 1 | ALA4266056 | cell-free format | Scientific Literature | |
| 19. | ALA4270260 | A | Fraction unbound in rhesus monkey plasma at 0.1 uM using [3H]-labeled compound | Macaca mulatta | 1 | ALA4266056 | cell-free format | Scientific Literature | |
| 20. | ALA4270261 | A | Clearance in rat at 1 mg/kg, iv or 2 mg/kg, po | Rattus norvegicus | 1 | ALA4266056 | organism-based format | Scientific Literature |
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