| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4255268 | B | Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes at 10 uM after 1 hr by microbeta scintillation counting method relative to control | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 2. | ALA4255269 | B | Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation counting method | Homo sapiens | 37 | cell-based format | Scientific Literature | ||
| 3. | ALA4255270 | B | Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes at 10 uM after 1 hr by microbeta scintillation counting method relative to control | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 4. | ALA4255273 | B | Displacement of [3H]CP55,940 from N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membranes after 1 hr by microbeta scintillation counting method | Homo sapiens | 37 | cell-based format | Scientific Literature | ||
| 5. | ALA4255274 | B | Selectivity ratio of Ki for N-terminal HA-tagged human CB2 receptor expressed in HEK293 cell membranes to Ki for N-terminal HA-tagged human CB1 receptor expressed in HEK293 cell membrane | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 6. | ALA4255276 | F | Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in forskolin-stimulated cAMP level by BRET assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA4255279 | F | Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in forskolin-stimulated cAMP level by BRET assay relative to control | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 8. | ALA4255281 | F | Agonist activity at N-terminal HA-tagged human CB1 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskolin-stimulated cAMP level by BRET assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 9. | ALA4255283 | F | Agonist activity at N-terminal HA-tagged human CB1 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskolin-stimulated cAMP level by BRET assay relative to control | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 10. | ALA4255286 | F | Inverse agonist activity at N-terminal HA-tagged human CB2 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as increase in forskolin-stimulated cAMP level at 10 uM by BRET assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 11. | ALA4255287 | F | Agonist activity at N-terminal HA-tagged human CB1 receptor expressed in HEK293 cells transfected with YFP-Epac-RLuc assessed as decrease in forskolin-stimulated cAMP level at 10 uM by BRET assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 12. | ALA4255289 | A | Effect on forskolin-stimulated cAMP level in HEK293 cells at 10 uM by BRET assay relative to control | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 13. | ALA4255290 | A | Effect on forskolin-stimulated cAMP level in HEK293 cells at 1 uM by BRET assay relative to control | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 14. | ALA4255291 | B | Inhibition of PCSK9 (unknown origin) | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 15. | ALA4255292 | F | Agonist activity at GPR120 (unknown origin) | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 16. | ALA4255293 | B | Inhibition of IL-17 (unknown origin) assessed as disruption of IL-17 protein-protein interaction | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 17. | ALA4255294 | F | Growth inhibition of Leishmania donovani | Leishmania donovani | 8 | organism-based format | Scientific Literature | ||
| 18. | ALA4255295 | B | Agonist activity at KCNQ2 (unknown origin) | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 19. | ALA4255296 | B | Agonist activity at KCNQ3 (unknown origin) | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 20. | ALA4255297 | B | Inhibition of NNMT (unknown origin) | Homo sapiens | 8 | single protein format | Scientific Literature |
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