| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4271527 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC1R expressed in HEK293 cells at 10 uM after 40 mins by gamma counting analysis relative to control | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 2. | ALA4271528 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting analysis | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 3. | ALA4271529 | F | Agonist activity at human MC1R expressed in HEK293 cells after 3 mins by cAMP assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 4. | ALA4271530 | F | Agonist activity at human MC1R expressed in HEK293 cells at 10 uM after 3 mins by cAMP assay relative to MT-2 | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 5. | ALA4271531 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting analysis | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 6. | ALA4271532 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC3R expressed in HEK293 cells at 10 uM after 40 mins by gamma counting analysis relative to control | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 7. | ALA4271533 | F | Agonist activity at human MC3R expressed in HEK293 cells after 3 mins by cAMP assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 8. | ALA4271534 | F | Agonist activity at human MC3R expressed in HEK293 cells at 10 uM after 3 mins by cAMP assay relative to MT-2 | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 9. | ALA4271535 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting analysis | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 10. | ALA4271536 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC4R expressed in HEK293 cells at 10 uM after 40 mins by gamma counting analysis relative to control | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 11. | ALA4271537 | F | Agonist activity at human MC4R expressed in HEK293 cells after 3 mins by cAMP assay | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 12. | ALA4271538 | F | Agonist activity at human MC4R expressed in HEK293 cells at 10 uM after 3 mins by cAMP assay relative to MT-2 | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 13. | ALA4271539 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting analysis | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 14. | ALA4271540 | B | Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC5R expressed in HEK293 cells at 10 uM after 40 mins by gamma counting analysis relative to control | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 15. | ALA4271541 | F | Agonist activity at human MC5R expressed in HEK293 cells after 3 mins by cAMP assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 16. | ALA4271542 | F | Agonist activity at human MC5R expressed in HEK293 cells at 10 uM after 3 mins by cAMP assay relative to MT-2 | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 17. | ALA4271543 | F | Induction of pigmentation effect in lizard at 3 ug/g, ip at 1 hr post dose | Anolis carolinensis | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA4271544 | B | Selectivity ratio of EC50 for human MC3R to EC50 for human MC1R | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4271545 | B | Selectivity ratio of EC50 for human MC4R to EC50 for human MC1R | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4271546 | B | Selectivity ratio of EC50 for human MC5R to EC50 for human MC1R | Homo sapiens | 1 | assay format | Scientific Literature |
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