| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4264824 | B | Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-Ala-Tyr) peptide as substrate after 5 mins in presence of ADP by fluorescence analysis | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 2. | ALA4264825 | B | Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide as substrate after 5 mins in presence of ADP by fluorescence analysis | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 3. | ALA4264826 | B | Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) peptide as substrate after 5 mins in presence of ADP by fluorescence analysis | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 4. | ALA4264827 | B | Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-Ala-Tyr) peptide as substrate after 1.5 hrs by ELISA | Homo sapiens | 15 | assay format | Scientific Literature | ||
| 5. | ALA4264828 | B | Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide as substrate after 1.5 hrs by ELISA | Homo sapiens | 15 | assay format | Scientific Literature | ||
| 6. | ALA4264829 | B | Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) peptide as substrate after 1.5 hrs by ELISA | Homo sapiens | 15 | assay format | Scientific Literature | ||
| 7. | ALA4264830 | B | Binding affinity to human wild type ABL1 (229 to 512 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 8. | ALA4264831 | B | Binding affinity to human wild type ABL1 (229 to 512 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 9. | ALA4264832 | B | Binding affinity to human wild type ABL1 (229 to 512 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 10 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 10. | ALA4264833 | B | Binding affinity to wild-type human partial length AURKA (E122 to K401 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 11. | ALA4264834 | B | Binding affinity to wild-type human partial length AURKA (E122 to K401 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 12. | ALA4264835 | B | Binding affinity to wild-type human partial length AURKA (E122 to K401 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 10 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 13. | ALA4264836 | B | Binding affinity to wild-type human partial length BRAF (S429 to E741 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 14. | ALA4264837 | B | Binding affinity to wild-type human partial length BRAF (S429 to E741 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 15. | ALA4264838 | B | Binding affinity to wild-type human partial length BRAF (S429 to E741 residues) expressed in mammalian expression system assessed as fraction of unbound kinase to substrate at 10 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 16. | ALA4264839 | B | Binding affinity to wild-type human full length CDK2 (M1 to L298 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 17. | ALA4264840 | B | Binding affinity to wild-type human full length CDK2 (M1 to L298 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 18. | ALA4264841 | B | Binding affinity to wild-type human full length CDK2 (M1 to L298 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 10 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 19. | ALA4264842 | B | Binding affinity to partial length wild type human EGFR (R669 to V1011 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 0.1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 20. | ALA4264843 | B | Binding affinity to partial length wild type human EGFR (R669 to V1011 residues) expressed in bacterial expression system assessed as fraction of unbound kinase to substrate at 1 uM after 1 hr by KinomeScan assay | Homo sapiens | 4 | assay format | Scientific Literature |
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