| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4266821 | B | Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) expressed in Escherichia coli BL21(DE3) after 1 hr by TopCount scintillation proximity assay | Homo sapiens | 28 | assay format | Scientific Literature | ||
| 2. | ALA4266822 | B | Displacement of [3H]-T0901317 from recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) expressed in Escherichia coli BL21(DE3) after 1 hr by scintillation proximity assay | Homo sapiens | 31 | assay format | Scientific Literature | ||
| 3. | ALA4266825 | B | Selectivity index, ratio of IC50 for recombinant human His-SUMO-tagged RORgamma LBD (265 to 518 residues) to IC50 for recombinant human His-SUMO-tagged RORbeta LBD (71 to 459 residues) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 4. | ALA4266826 | B | Inverse agonist activity at GAL4-DNA binding domain-fused human RORbeta ligand binding domain expressed in HEK293T cells incubated for 20 hrs by luciferase reporter gene assay | Homo sapiens | 3 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!