| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3755536 | B | Displacement of 125I-labeled [Nle4,DPhe7]-alpha-MSH from human melanocortin 3 receptor expressed in HEK293 cells incubated for 40 mins by gamma counting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 2. | ALA3755537 | B | Displacement of 125I-labeled [Nle4,DPhe7]-alpha-MSH from human melanocortin 4 receptor expressed in HEK293 cells incubated for 40 mins by gamma counting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 3. | ALA3755538 | B | Displacement of 125I-labeled [Nle4,DPhe7]-alpha-MSH from human melanocortin 5 receptor expressed in HEK293 cells incubated for 40 mins by gamma counting analysis | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA3755539 | F | Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as intracellular cAMP accumulation incubated for 3 mins in presence of IBMX | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 5. | ALA3755540 | F | Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as intracellular cAMP accumulation incubated for 3 mins in presence of IBMX | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 6. | ALA3755541 | F | Agonist activity at human melanocortin 4 receptor expressed in HEK293 cells assessed as intracellular cAMP accumulation incubated for 3 mins in presence of IBMX | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 7. | ALA3755542 | F | Agonist activity at human melanocortin 5 receptor expressed in HEK293 cells assessed as intracellular cAMP accumulation incubated for 3 mins in presence of IBMX | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 8. | ALA3755543 | B | Displacement of 125I-labeled [Nle4,DPhe7]-alpha-MSH from human melanocortin 1 receptor expressed in HEK293 cells at 10 uM incubated for 40 mins by gamma counting analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA3755544 | F | Agonist activity at human melanocortin 1 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation incubated for 3 mins relative to MT-2 | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 10. | ALA3755545 | F | Agonist activity at human melanocortin 3 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation incubated for 3 mins relative to MT-2 | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 11. | ALA3755547 | F | Agonist activity at human melanocortin 5 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation incubated for 3 mins relative to MT-2 | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 12. | ALA3755737 | B | Selectivity ratio of EC50 for human melanocortin 4 receptor expressed in HEK293 cells to EC50 for human melanocortin 3 receptor expressed in HEK293 cells | Homo sapiens | 1 | cell-based format | Scientific Literature |
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