# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4406751 | B | Inhibition of human ALK2 using casein as substrate in presence of 10 uM [gamma33P] ATP by radioactive assay | Homo sapiens | 25 | ALA4402613 | single protein format | Scientific Literature | |
2. | ALA4406752 | A | Inhibition of human ALK5 using casein as substrate in presence of 10 uM [gamma33P] ATP by radioactive assay | Homo sapiens | 25 | ALA4402613 | single protein format | Scientific Literature | |
3. | ALA4406753 | B | Selectivity index, ratio of IC50 for inhibition of human ALK5 using casein as substrate in presence of 10 uM [gamma33P] ATP by radioactive assay to IC50 for inhibition of human ALK3 using casein as substrate in presence of 10 uM [gamma33P] ATP by radioactive assay | Homo sapiens | 20 | ALA4402613 | assay format | Scientific Literature | |
4. | ALA4406758 | B | Inhibition of C-terminal nanoluciferase-fused ALK2 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by NanoBRET NanoGlo Substrate addition by NanoBRET assay | Homo sapiens | 21 | ALA4402613 | cell-based format | Scientific Literature | |
5. | ALA4406759 | A | Inhibition of ALK5 (unknown origin) expressed in HEK293 cells transfected with CAGA-luciferase and Renilla luciferase reporter measured after 24 hrs by dual luciferase reporter assay | Homo sapiens | 21 | ALA4402613 | cell-based format | Scientific Literature | |
6. | ALA4406760 | U | Selectivity index, ratio of IC50 for inhibition of ALK5 (unknown origin) expressed in HEK293 cells transfected with CAGA-luciferase and Renilla luciferase reporter measured after 24 hrs by dual luciferase reporter assay to IC50 for inhibition of C-terminal nanoluciferase-fused ALK2 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by NanoBRET NanoGlo Substrate addition by NanoBRET assay | Homo sapiens | 18 | ALA4402613 | cell-based format | Scientific Literature | |
7. | ALA4406761 | A | Apparent permeability across apical to basolateral membrane in human Caco2 cells at 5 uM incubated for 120 mins in orbital shaker by LC-QTOF/MS analysis | Homo sapiens | 4 | ALA4402613 | cell-based format | Scientific Literature | |
8. | ALA4406762 | A | Apparent permeability across basolateral to apical membrane in human Caco2 cells at 5 uM incubated for 120 mins in orbital shaker by LC-QTOF/MS analysis | Homo sapiens | 4 | ALA4402613 | cell-based format | Scientific Literature | |
9. | ALA4406763 | A | Efflux ratio of apparent permeability across basolateral to apical membrane over apical to basolateral membrane in human Caco2 cells at 5 uM incubated for 120 mins in orbital shaker by LC-QTOF/MS analysis | Homo sapiens | 4 | ALA4402613 | cell-based format | Scientific Literature | |
10. | ALA4406769 | B | Inhibition of human ERG expressed in HEK293 cells measured after 5 mins by whole cell patch clamp method | Homo sapiens | 3 | ALA4402613 | cell-based format | Scientific Literature | |
11. | ALA4406770 | B | Inhibition of ALK1 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
12. | ALA4406771 | B | Inhibition of ALK2 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
13. | ALA4406772 | B | Inhibition of ALK3 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
14. | ALA4406773 | B | Inhibition of ALK6 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
15. | ALA4406774 | B | Inhibition of ARAF (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
16. | ALA4406775 | B | Inhibition of MAP4K4 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
17. | ALA4406776 | B | Inhibition of MINK (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
18. | ALA4406777 | B | Inhibition of TNK1 (unknown origin) at 1 uM | Homo sapiens | 3 | ALA4402613 | single protein format | Scientific Literature | |
19. | ALA4406778 | A | Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate incubated for 40 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 3 | ALA4402613 | microsome format | Scientific Literature | |
20. | ALA4406779 | A | Inhibition of CYP2B6 in human liver microsomes using bupropion as substrate incubated for 40 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 3 | ALA4402613 | microsome format | Scientific Literature |
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