| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4310221 | B | Inhibition of recombinant His-tagged TAF1 bromodomain 2 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 2. | ALA4310222 | B | Inhibition of recombinant His-tagged TAF1 bromodomain 1 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 3. | ALA4310223 | B | Inhibition of recombinant His-tagged BRD4 bromodomain 1 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 4. | ALA4310224 | B | Inhibition of recombinant His-tagged BRD4 bromodomain 2 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 5. | ALA4310225 | B | Inhibition of recombinant His-tagged BRD9 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 6. | ALA4310226 | B | Inhibition of recombinant His-tagged CECR2 (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 27 | single protein format | Scientific Literature | ||
| 7. | ALA4310227 | B | Inhibition of recombinant His-tagged CBP (unknown origin) after 10 mins by TR-FRET assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 8. | ALA4425846 | B | Inhibition of recombinant His-tagged BRD4 bromodomain1 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 9. | ALA4425847 | B | Inhibition of recombinant His-tagged BRD4 bromodomain2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 10. | ALA4425848 | B | Displacement of biotinylated JQ1 analog from recombinant His-tagged CBP (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 11. | ALA4425849 | B | Displacement of biotinylated JQ1 analog from recombinant His-tagged BRPF1 (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 12. | ALA4425850 | B | Displacement of biotinylated JQ1 analog from recombinant His-tagged BRD9 (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 13. | ALA4425851 | B | Inhibition of recombinant His-tagged TAF1 isoform-1 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 14. | ALA4425852 | B | Inhibition of recombinant His-tagged TAF1 isoform-2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 15. | ALA4425853 | B | Inhibition of recombinant His-tagged CECR2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 16. | ALA4425854 | B | Selectivity index, ratio of IC50 for recombinant His-tagged BRD9 (unknown origin) to IC50 for recombinant His-tagged TAF1 isoform-2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4425855 | B | Selectivity index, ratio of IC50 for recombinant His-tagged BRD4 to IC50 for recombinant His-tagged TAF1 isoform-2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4425862 | B | Binding affinity to wild type BRD9 (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 19. | ALA4425863 | B | Binding affinity to BRD9 Y106I mutant (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 20. | ALA4425864 | B | Binding affinity to BRD9 M92I mutant (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | single protein format | Scientific Literature |
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