| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4408783 | Binding | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) | Homo sapiens | 5 | ALA4406837 | protein complex format | Scientific Literature | |
| 2. | ALA4408794 | Binding | Competitive irreversible inhibition of CDK12/cyclinK (unknown origin) in presence of Km ATP | Homo sapiens | 5 | ALA4406837 | protein complex format | Scientific Literature | |
| 3. | ALA4408796 | Binding | Competitive irreversible inhibition of CDK9/cyclin T (unknown origin) in presence of Km ATP | Homo sapiens | 5 | ALA4406837 | protein complex format | Scientific Literature | |
| 4. | ALA4408801 | Binding | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) assessed as inactivation constant using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate | Homo sapiens | 4 | ALA4406837 | protein complex format | Scientific Literature | |
| 5. | ALA4408802 | Binding | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate | Homo sapiens | 4 | ALA4406837 | protein complex format | Scientific Literature | |
| 6. | ALA4408803 | Binding | Ratio of Ki CDK7/cyclinH/MAT1 (unknown origin) to Kinact CDK7/cyclinH/MAT1 (unknown origin) assessed as inactivation constant | Homo sapiens | 4 | ALA4406837 | protein complex format | Scientific Literature | |
| 7. | ALA4408804 | Functional | Antiproliferative activity against human HL60 cells after 72 hrs by CellTiter-Glo assay | Homo sapiens | 4 | ALA4406837 | cell-based format | Scientific Literature | |
| 8. | ALA4408805 | ADME | Clearance in mouse | Mus musculus | 4 | ALA4406837 | organism-based format | Scientific Literature | |
| 9. | ALA4408806 | Binding | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of Km ATP | Homo sapiens | 4 | ALA4406837 | protein complex format | Scientific Literature | |
| 10. | ALA4408807 | Binding | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of 2 mM ATP | Homo sapiens | 4 | ALA4406837 | protein complex format | Scientific Literature | |
| 11. | ALA4611856 | ADME | Clearance in mouse plasma by LC/MS-MS analysis | Mus musculus | 4 | ALA4610077 | cell-free format | Scientific Literature | |
| 12. | ALA4611857 | Binding | Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP addition | Homo sapiens | 9 | ALA4610077 | protein complex format | Scientific Literature |
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