| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4428988 | B | Inhibition of human recombinant AKR1C3 using S-tetralol as substrate assessed as reduction in NADP+-dependent S-tetralol oxidation preincubated for 10 mins followed by protein addition by fluorometric assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 2. | ALA4428989 | B | Inhibition of human recombinant AKR1C2 using S-tetralol as substrate assessed as reduction in NADP+-dependent S-tetralol oxidation preincubated for 10 mins followed by protein addition by fluorometric assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 3. | ALA4428990 | B | Selectivity ratio of IC50 for human recombinant AKR1C2 to IC50 for human recombinant AKR1C3 | Homo sapiens | 14 | assay format | Scientific Literature | ||
| 4. | ALA4429007 | B | Inhibition of COX2 (unknown origin) using arachidonic acid as substrate assessed as reduction in PGH2 conversion to PGG2 by measuring TMPD oxidation at 10 uM preincubated for 5 mins followed by substrate/TMPD addition measured for 5 mins by colorimetric assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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