| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4407669 | B | Inhibition of GST-tagged recombinant human DDR1 (440 to 876 amino acids) expressed in baculovirus using fluorescein-poly GAT as substrate after 1 hr by FRET-based LanthaScreen Eu kinase binding assay | Homo sapiens | 15 | ALA4406813 | assay format | Scientific Literature | |
| 2. | ALA4407670 | A | Inhibition of GST-tagged recombinant human DDR2 expressed in baculovirus using fluorescein-poly GAT as substrate after 1 hr by FRET-based LanthaScreen Eu kinase binding assay | Homo sapiens | 15 | ALA4406813 | assay format | Scientific Literature | |
| 3. | ALA4407671 | A | Inhibition of His-tagged human TrkA expressed in baculovirus expression system using Tyr1 peptide as substrate after 1.5 hrs by FRET-based Z-LYTE assay | Homo sapiens | 15 | ALA4406813 | assay format | Scientific Literature | |
| 4. | ALA4407672 | A | Inhibition of His-tagged human TrkB expressed in baculovirus expression system using Tyr1 peptide as substrate after 1.5 hrs by FRET-based Z-LYTE assay | Homo sapiens | 15 | ALA4406813 | assay format | Scientific Literature | |
| 5. | ALA4407673 | A | Inhibition of His-tagged human TrkC expressed in baculovirus expression system using Tyr1 peptide as substrate after 1.5 hrs by FRET-based Z-LYTE assay | Homo sapiens | 15 | ALA4406813 | assay format | Scientific Literature | |
| 6. | ALA4407674 | B | Binding affinity to wild-type human partial length DDR1 (R565 to V876 residues) expressed in bacterial expression system | Homo sapiens | 1 | ALA4406813 | assay format | Scientific Literature | |
| 7. | ALA4407675 | A | Inhibition of wild-type human partial length DDR2 (V555 to E855 residues) expressed in HEK-293 cells at 1 uM after 1 hr by quantitative PCR based KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 8. | ALA4407676 | A | Inhibition of wild-type human ABL1 (S229 to K512 residues) expressed in HEK-293 cells at 1 uM after 1 hr by quantitative PCR based KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 9. | ALA4407677 | A | Inhibition of wild-type human partial length KIT (I571 to D952 residues) expressed in Escherichia coli BL21 at 1 uM after 1 hr by quantitative PCR based KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4406813 | assay format | Scientific Literature | |
| 10. | ALA4407678 | A | Inhibition of wild-type human partial length PDGFRB (V582 to Y1009 residues) expressed in Escherichia coli BL21 at 1 uM after 1 hr by quantitative PCR based KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4406813 | assay format | Scientific Literature | |
| 11. | ALA4407679 | A | Inhibition of wild-type human partial length TRKC (Q531 to G825 residues) expressed in HEK-293 cells at 1 uM after 1 hr by quantitative PCR based KINOMEscan assay relative to control | Homo sapiens | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 12. | ALA4407680 | A | Inhibition of human DDR2 | Homo sapiens | 1 | ALA4406813 | single protein format | Scientific Literature | |
| 13. | ALA4407681 | A | Inhibition of human ABL1 | Homo sapiens | 1 | ALA4406813 | single protein format | Scientific Literature | |
| 14. | ALA4407682 | A | Inhibition of human KIT | Homo sapiens | 1 | ALA4406813 | single protein format | Scientific Literature | |
| 15. | ALA4407683 | A | Inhibition of human PDGFRB | Homo sapiens | 1 | ALA4406813 | single protein format | Scientific Literature | |
| 16. | ALA4407684 | A | Inhibition of human TrkC | Homo sapiens | 1 | ALA4406813 | single protein format | Scientific Literature | |
| 17. | ALA4407685 | B | Inhibition of DDR1 in mouse Pan02 cells assessed as reduction in collagen-induced DDR1 phosphorylation after 8 hrs by Western blot analysis | Mus musculus | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 18. | ALA4407686 | B | Inhibition of DDR1 in mouse Pan02 cells assessed as reduction in collagen-induced PYK2 phosphorylation after 8 hrs by Western blot analysis | Mus musculus | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 19. | ALA4407687 | B | Inhibition of DDR1 in mouse Pan02 cells assessed as reduction in collagen-induced PEAK1 phosphorylation after 8 hrs by Western blot analysis | Mus musculus | 1 | ALA4406813 | cell-based format | Scientific Literature | |
| 20. | ALA4407688 | B | Inhibition of DDR1 in mouse Pan02 cells assessed as reduction in epithelial-mesenchymal transition by measuring down regulation of collagen-induced N-Cadherin expression at 1 uM incubated for 24 hrs by DAPI staining based immunofluorescence method | Mus musculus | 1 | ALA4406813 | cell-based format | Scientific Literature |
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