# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4379074 | B | Inhibition of human PKA using Kemptide as substrate incubated for 40 mins in presence of [gamma-33P]ATP by radiometric scintillation counting analysis | Homo sapiens | 57 | ALA4376834 | assay format | Scientific Literature | |
2. | ALA4379075 | B | Inhibition of recombinant human ROCK1 (17 to 535 residues) using KEAKEKRQEQIAKR as substrate incubated for 40 mins in presence of [gamma-33P]ATP and 10 uM ATP by radiometric scintillation counting analysis | Homo sapiens | 57 | ALA4376834 | single protein format | Scientific Literature | |
3. | ALA4379076 | B | Inhibition of recombinant human ROCK2 (11 to 552 residues) using KEAKEKRQEQIAKR as substrate incubated for 40 mins in presence of [gamma-33P]ATP and 10 uM ATP by radiometric scintillation counting analysis | Homo sapiens | 57 | ALA4376834 | single protein format | Scientific Literature | |
4. | ALA4379077 | B | Inhibition of human LIMK2 in presence of 10 uM of ATP by radiometric analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
5. | ALA4379078 | B | Inhibition of human recombinant full length AURORA-A I31F mutant using kemptide as substrate incubated for 40 mins in presence of [gamma-33P]ATPand 10 uM ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | assay format | Scientific Literature | |
6. | ALA4379079 | B | Inhibition of recombinant full length human AURORA-B using AKRRRLSSLRA as substrate incubated for 40 mins in presence of [gamma-33P]ATP and 10 uM ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
7. | ALA4379080 | B | Inhibition of recombinant full length human PKG1alpha using RRRLSFAEPG as substrate incubated for 40 mins in presence of [gamma-33P]ATP and 10 uM ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
8. | ALA4379081 | B | Inhibition of recombinant full length human PKG1beta using RRRLSFAEPG as substrate incubated for 40 mins in presence of [gamma-33P]ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
9. | ALA4379082 | B | Binding affinity to DNMT2 (unknown origin) at protein to compound concentration ratio of 1:20 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
10. | ALA4379083 | B | Binding affinity to NSD2 (unknown origin) at protein to compound concentration ratio of 1:20 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
11. | ALA4379084 | B | Binding affinity to TRIM24 (unknown origin) at protein to compound concentration ratio of 1:10 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
12. | ALA4379085 | B | Binding affinity to SETDB1 (unknown origin) at protein to compound concentration ratio of 1:10 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
13. | ALA4379086 | B | Binding affinity to WTAP (unknown origin) at protein to compound concentration ratio of 1:20 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
14. | ALA4379087 | B | Binding affinity to STING (unknown origin) at protein to compound concentration ratio of 1:10 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
15. | ALA4379088 | B | Binding affinity to JMJD5 (unknown origin) at protein to compound concentration ratio of 1:10 by differential scanning fluorimetry | Homo sapiens | 1 | ALA4376834 | single protein format | Scientific Literature | |
16. | ALA4379089 | F | Antiproliferative activity against human PANC1 cells assessed as reduction in cell viability | Homo sapiens | 1 | ALA4376834 | cell-based format | Scientific Literature | |
17. | ALA4379090 | F | Antiproliferative activity against human MIAPaCa2 cells assessed as reduction in cell viability | Homo sapiens | 1 | ALA4376834 | cell-based format | Scientific Literature | |
18. | ALA4379091 | F | Antiproliferative activity against human AsPC1 assessed as reduction in cell viability | Homo sapiens | 1 | ALA4376834 | cell-based format | Scientific Literature | |
19. | ALA4379092 | F | Antiproliferative activity against human BxPC1 cells assessed as reduction in cell viability | Homo sapiens | 1 | ALA4376834 | cell-based format | Scientific Literature | |
20. | ALA4379093 | F | Antiproliferative activity against human OCUT-2C cells assessed as reduction in cell viability | Homo sapiens | 1 | ALA4376834 | cell-based format | Scientific Literature |