#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4421913	B	Inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as residual enzyme activity for geranylgeranylation of K-Ras4B at 50 uM incubated for 30 mins in presence of [3H]GGPP by scintillation counting assay relative to control	Rattus norvegicus	701		assay format	Patent Bioactivity Data
2.	ALA4421914	B	Inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as residual enzyme activity for geranylgeranylation of RhoA at 50 uM incubated for 30 mins in presence of [3H]GGPP by scintillation counting assay relative to control	Rattus norvegicus	128		assay format	Patent Bioactivity Data
3.	ALA4421915	B	Inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of K-Ras4B incubated for 30 mins in presence of [3H]GGPP by scintillation counting assay	Rattus norvegicus	13		assay format	Patent Bioactivity Data
4.	ALA4421916	B	Inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of RhoA incubated for 30 mins in presence of [3H]GGPP by scintillation counting assay relative to control	Rattus norvegicus	87		assay format	Patent Bioactivity Data
5.	ALA4421917	F	Antiproliferative activity against human K562 cells assessed as inhibition of cell proliferation incubated for 72 hrs by CCK8 assay	Homo sapiens	27		cell-based format	Patent Bioactivity Data
6.	ALA4421920	F	Antiproliferative activity against human Jurkat cells assessed as inhibition of cell proliferation incubated for 72 hrs by CCK8 assay	Homo sapiens	33		cell-based format	Patent Bioactivity Data
7.	ALA4421930	B	Competitive inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of RhoA incubated for 30 mins in presence of fixed level of [3H]GGPP and varying RhoA levels by scintillation counting assay relative to control	Rattus norvegicus	2		assay format	Patent Bioactivity Data
8.	ALA4421931	B	Competitive inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of RhoA incubated for 30 mins in presence of varying level of [3H]GGPP and fixed RhoA levels by scintillation counting assay relative to control	Rattus norvegicus	4		assay format	Patent Bioactivity Data
9.	ALA4421932	B	Inhibition of geranylgeranyltransferase type I in HEK293 cells expressing Myc-HA-tagged Rheb-WT assessed as effect on unprenylated Rap1 accumulation at 3.1 to 25 uM incubated for 48 hrs by SDS-PAGE and immunoblot analysis	Homo sapiens	2		cell-based format	Patent Bioactivity Data
10.	ALA4421933	B	Inhibition of geranylgeranyltransferase type I in HEK293 cells expressing Myc-HA-tagged Rheb-CVSL assessed as effect on unprenylated Rap1 accumulation at 12.5 to 50 uM incubated for 48 hrs by SDS-PAGE and immunoblot analysis	Homo sapiens	2		cell-based format	Patent Bioactivity Data
11.	ALA4421937	F	Antiproliferative activity against human Jurkat cells assessed as inhibition of cell proliferation at 12.5 uM incubated for 72 hrs by CCK8 assay	Homo sapiens	1		cell-based format	Patent Bioactivity Data
12.	ALA4421938	F	Antiproliferative activity against human PANC1 cells assessed as inhibition of cell proliferation at 12.5 uM incubated for 72 hrs by CCK8 assay	Homo sapiens	1		cell-based format	Patent Bioactivity Data
13.	ALA4421939	B	Inhibition of RabGGTase (unknown origin) up to 10000 nM using YPTI as substrate protein and [3H]geranylgeranyl pyrophosphate incubated for 20 mins by scintillation counting assay	Homo sapiens	1		protein complex format	Patent Bioactivity Data
14.	ALA4421941	B	Inhibition of rat recombinant FTase alpha/beta expressed in Escherichia coli at 50000 nM using K-Ras4B as a substrate as and [3H]farnesyl pyrophosphate incubated for 30 mins by scintillation counting assay	Rattus norvegicus	2		assay format	Patent Bioactivity Data
15.	ALA4421942	B	Uncompetitive inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of RhoA incubated for 30 mins in presence of varying level of [3H]GGPP and fixed RhoA levels by scintillation counting assay by Michaelis-Menten plot analysis	Rattus norvegicus	2		assay format	Patent Bioactivity Data
16.	ALA4421943	B	Competitive inhibition of rat recombinant geranylgeranyltransferase type I expressed in Escherichia coli assessed as reduction in geranylgeranylation of RhoA incubated for 30 mins in presence of fixed level of [3H]GGPP and varying RhoA levels by scintillation counting assay by Michaelis-Menten plot analysis	Rattus norvegicus	2		assay format	Patent Bioactivity Data
17.	ALA4421944	B	Inhibition of geranylgeranyltransferase type I in HEK293 cells expressing Myc-HA-tagged Rheb-WT assessed as effect on unprenylated Rap1 accumulation at 2.5 uM incubated for 48 hrs by SDS-PAGE and immunoblot analysis	Homo sapiens	2		cell-based format	Patent Bioactivity Data