# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4372182 | B | Inhibition of bovine cationic trypsin using Bz-FVR-pNA as substrate after 30 mins | Bos taurus | 3 | single protein format | Scientific Literature | ||
2. | ALA4372183 | B | Inhibition of human plasmin using Ac-RM(O2)YR-pNA as substrate after 30 mins | Homo sapiens | 18 | single protein format | Scientific Literature | ||
3. | ALA4372185 | B | Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 mins | Homo sapiens | 3 | single protein format | Scientific Literature | ||
4. | ALA4372190 | B | Inhibition of activated beta-factor 9 (unknown origin) using Boc-QGR-MCA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
5. | ALA4372191 | B | Inhibition of activated factor 10 (unknown origin) using Ac-QRSR-pNA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
6. | ALA4372192 | B | Inhibition of activated beta-factor 12 (unknown origin) using Ac-QRFR-pNA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
7. | ALA4372193 | B | Inhibition of human thrombin using Ac-ATPR-pNA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
8. | ALA4372194 | B | Inhibition of tPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
9. | ALA4372195 | B | Inhibition of uPA (unknown origin) using Z-Pyr-Gly-Arg-MCA as substrate after 30 mins relative to untreated control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
10. | ALA4372196 | B | Inhibition of activated beta-factor 11 (unknown origin) using Bz-FVRpNA as substrate after 30 mins relative to untreated control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
11. | ALA4372197 | B | Inhibition of plasma KLK (unknown origin) using Ac-NLTR-pNA as substrate after 30 mins relative to untreated control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
12. | ALA4372198 | B | Inhibition of matriptase (unknown origin) using Boc-QAR-MCA as substrate after 30 mins relative to untreated control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
13. | ALA4372199 | B | Inhibition of human plasmin assessed as dissociation rate constant using Ac-RM(O2)YR-pNA as substrate after 30 mins | Homo sapiens | 1 | single protein format | Scientific Literature | ||
14. | ALA4372200 | B | Inhibition of human plasmin assessed as association rate constant using Ac-RM(O2)YR-pNA as substrate after 30 mins | Homo sapiens | 1 | single protein format | Scientific Literature | ||
15. | ALA4372203 | B | Inhibition of plasmin in human plasma assessed as reduction in tPA and thrombin-induced fibrinolysis at 400 nM by fibrin light scattering analysis relative to control | Homo sapiens | 1 | cell-free format | Scientific Literature | ||
16. | ALA4372204 | B | Inhibition of plasmin in human plasma assessed as reduction in tPA and thrombin-induced fibrinolysis at 200 nM by fibrin light scattering analysis relative to control | Homo sapiens | 1 | cell-free format | Scientific Literature | ||
17. | ALA4372207 | B | Selectivity index, ratio of IC50 for inhibition of activated beta-factor 9 (unknown origin) to IC50 for Inhibition of human plasmin | Homo sapiens | 1 | assay format | Scientific Literature | ||
18. | ALA4372208 | B | Selectivity index, ratio of IC50 for inhibition of activated factor 10 (unknown origin) to IC50 for Inhibition of human plasmin | Homo sapiens | 1 | assay format | Scientific Literature | ||
19. | ALA4372209 | B | Selectivity index, ratio of IC50 for inhibition of activated beta-factor 12 (unknown origin) to IC50 for Inhibition of human plasmin | Homo sapiens | 1 | assay format | Scientific Literature | ||
20. | ALA4372210 | B | Selectivity index, ratio of IC50 for inhibition of human thrombin to IC50 for Inhibition of human plasmin | Homo sapiens | 1 | assay format | Scientific Literature |