| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4408783 | B | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) | Homo sapiens | 5 | protein complex format | Scientific Literature | ||
| 2. | ALA4408794 | B | Competitive irreversible inhibition of CDK12/cyclinK (unknown origin) in presence of Km ATP | Homo sapiens | 5 | protein complex format | Scientific Literature | ||
| 3. | ALA4408796 | B | Competitive irreversible inhibition of CDK9/cyclin T (unknown origin) in presence of Km ATP | Homo sapiens | 5 | protein complex format | Scientific Literature | ||
| 4. | ALA4408801 | B | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) assessed as inactivation constant using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 5. | ALA4408802 | B | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 6. | ALA4408803 | B | Ratio of Ki CDK7/cyclinH/MAT1 (unknown origin) to Kinact CDK7/cyclinH/MAT1 (unknown origin) assessed as inactivation constant | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 7. | ALA4408804 | F | Antiproliferative activity against human HL60 cells after 72 hrs by CellTiter-Glo assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 8. | ALA4408805 | A | Clearance in mouse | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 9. | ALA4408806 | B | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of Km ATP | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 10. | ALA4408807 | B | Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of 2 mM ATP | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 11. | ALA4611856 | A | Clearance in mouse plasma by LC/MS-MS analysis | Mus musculus | 4 | cell-free format | Scientific Literature | ||
| 12. | ALA4611857 | B | Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP addition | Homo sapiens | 9 | protein complex format | Scientific Literature |
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