# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4415166 | B | Inhibition of DYRK1A (unknown origin) by TR-FRET assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
2. | ALA4415167 | B | Inhibition of DYRK1A (unknown origin) by ADP assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
3. | ALA4415168 | B | Inhibition of CLK1 (unknown origin) by TR-FRET assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
4. | ALA4415172 | F | Inhibition of DYRK1A in mouse at 3 mg/kg relative to control | Mus musculus | 2 | organism-based format | Scientific Literature | ||
5. | ALA5251363 | B | Inhibition of recombinant human CDK5/p25 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
6. | ALA5251364 | B | Inhibition of recombinant human CK1epsilon expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
7. | ALA5251365 | B | Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
8. | ALA5251366 | B | Inhibition of recombinant human CLK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
9. | ALA5251367 | B | Inhibition of recombinant human CLK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
10. | ALA5251368 | B | Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
11. | ALA5251369 | B | Inhibition of recombinant human DYRK1A expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
12. | ALA5251370 | B | Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
13. | ALA5251371 | B | Inhibition of recombinant human DYRK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
14. | ALA5251372 | B | Inhibition of recombinant human DYRK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
15. | ALA5251373 | B | Inhibition of recombinant human DYRK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
16. | ALA5251374 | B | Inhibition of recombinant human GSK-3beta expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
17. | ALA5251375 | B | Selectivity ratio of IC50 for recombinant human CLK1 expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 46 | cell-based format | Scientific Literature | ||
18. | ALA5251376 | B | Selectivity ratio of IC50 for recombinant human DYRK1B expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 48 | cell-based format | Scientific Literature | ||
19. | ALA5251377 | B | Selectivity ratio of IC50 for recombinant human GSK-3beta expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 48 | cell-based format | Scientific Literature | ||
20. | ALA5251378 | B | Inhibition of recombinant human CLK1 expressed in Sf9 insect cells using myelin basic protein as substrate incubated for 110 mins in presence of ATP by non-radioactive ADP-Glo luminescence microplate reader assay | Homo sapiens | 35 | cell-based format | Scientific Literature |