| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4413958 | B | Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 11 | ALA4411328 | single protein format | Scientific Literature | |
| 2. | ALA4413959 | B | Inhibition of human CPA2 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 11 | ALA4411328 | single protein format | Scientific Literature | |
| 3. | ALA4413960 | B | Inhibition of human CPA4 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 11 | ALA4411328 | single protein format | Scientific Literature | |
| 4. | ALA4413962 | B | Inhibition of human CPA1 using AAFP as substrate assessed as dissociation rate constant measured at pre-steady state by spectrophotometry | Homo sapiens | 4 | ALA4411328 | single protein format | Scientific Literature | |
| 5. | ALA4413963 | B | Inhibition of human CPA1 using AAFP as substrate assessed as apparent first-order rate constant measured at pre-steady state by measuring Koff/Kon ratio by spectrophotometry | Homo sapiens | 4 | ALA4411328 | single protein format | Scientific Literature | |
| 6. | ALA4413964 | B | Inhibition of human CPA1 using AAFP as substrate assessed as association rate constant measured at pre-steady state by spectrophotometry | Homo sapiens | 4 | ALA4411328 | single protein format | Scientific Literature | |
| 7. | ALA4413965 | B | Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometry | Homo sapiens | 4 | ALA4411328 | single protein format | Scientific Literature | |
| 8. | ALA4413966 | B | Inhibition of human CPD at 1 nM to 1 mM using AAFA as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 11 | ALA4411328 | single protein format | Scientific Literature | |
| 9. | ALA4413967 | B | Inhibition of human CPB1 at 1 nM to 1 mM using AAFA as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 10 | ALA4411328 | single protein format | Scientific Literature | |
| 10. | ALA4413968 | B | Inhibition of rat CPA3 using AAFP as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Rattus norvegicus | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 11. | ALA4413969 | B | Inhibition of human TAFI at 1 nM to 1 mM using AAFA as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 12. | ALA4413970 | B | Inhibition of human CPN at 1 nM to 1 mM using N-(3-[2-furyl]acryloyl)-alanyl-lysine-OH as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 13. | ALA4413971 | B | Inhibition of human CCP1 at 1 nM to mM using tubulin as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 14. | ALA4413972 | B | Inhibition of human CCP6 at 1 nM to 1 mM using tubulin as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 15. | ALA4413973 | B | Inhibition of human MMP9 using fluorogenic Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 peptide as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 16. | ALA4413974 | A | Drug uptake in CPA3 expressing human HeLa cells at 1 to 5 uM treated for 6 hrs followed by cell wash and measured by DAPI-staining based fluorescence confocal microscopy | Homo sapiens | 1 | ALA4411328 | cell-based format | Scientific Literature | |
| 17. | ALA4413975 | B | Inhibition of human MMP10 using fluorogenic Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 peptide as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 18. | ALA4413976 | B | Inhibition of human MMP12 using fluorogenic Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 peptide as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 19. | ALA4413977 | B | Inhibition of human MMP13 using fluorogenic Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 peptide as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature | |
| 20. | ALA4413981 | B | Inhibition of human neutrophil Elastase at 1 nM to 1 mM using succinyl-alanylalanyl-prolyl-valine-4-nitroanilide as substrate preincubated for 45 mins measured at 30 sec intervals for 15 mins by UV/vis-spectrophotometry | Homo sapiens | 1 | ALA4411328 | single protein format | Scientific Literature |
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