# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4345228 | B | Inhibition of PI5P4Kalpha (unknown origin) incubated for 15 mins in presence of ATP by ADP-Glo assay | Homo sapiens | 18 | ALA4342488 | single protein format | Scientific Literature | |
2. | ALA4345229 | B | Inhibition of PI5P4Kbeta (unknown origin) incubated for 15 mins in presence of ATP by ADP-Glo assay | Homo sapiens | 17 | ALA4342488 | single protein format | Scientific Literature | |
3. | ALA4345230 | B | Inhibition of human MSK2 expressed in bacteria assessed as enzyme activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4342488 | assay format | Scientific Literature | |
4. | ALA4345231 | B | Inhibition of human TYK2 expressed in mammalian expression system assessed as enzyme activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4342488 | assay format | Scientific Literature | |
5. | ALA4345232 | B | Inhibition of wild-type human full length CSNK2A2 (M1 to R350 residues) expressed in mammalian expression system assessed as enzyme activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4342488 | assay format | Scientific Literature | |
6. | ALA4345233 | B | Inhibition of wild-type human partial length PDGFRB (V582 to Y1009 residues) expressed in bacterial expression system assessed as enzyme activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4342488 | assay format | Scientific Literature | |
7. | ALA4345234 | B | Inhibition of wild-type human partial length PIKFYVE (F1512 to C2098 residues) expressed in mammalian expression system assessed as enzyme activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4342488 | assay format | Scientific Literature | |
8. | ALA4345235 | B | Induction of stabilization of PI5P4Kalpha in HEK293T cells at 10 uM incubated for 1 hr at 58 to 61 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 1 | ALA4342488 | cell-based format | Scientific Literature | |
9. | ALA4345236 | B | Induction of stabilization of PI5P4Kbeta in HEK293T cells at 10 uM incubated for 1 hr at 58 to 61 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 1 | ALA4342488 | cell-based format | Scientific Literature | |
10. | ALA4345237 | B | Binding affinity to PI5P4Kalpha in HEK293T cells at 1 to 10 uM incubated for 1 hr at 52 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 4 | ALA4342488 | cell-based format | Scientific Literature | |
11. | ALA4345238 | B | Binding affinity to PI5P4Kbeta in HEK293T cells at 1 to 10 uM incubated for 1 hr at 52 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 4 | ALA4342488 | cell-based format | Scientific Literature | |
12. | ALA4345239 | B | Inhibition of N-terminal GST-tagged full length human PIKFYVE (1 to 2098 residues) using PI(3)P and Phosphatidylserine as substrate by ADP-Glo assay | Homo sapiens | 1 | ALA4342488 | single protein format | Scientific Literature | |
13. | ALA4406331 | B | Binding affinity to recombinant PI5P4Kalpha (unknown origin) assessed as protein-labeling at 10 uM incubated for 2 hrs by mass spectrometry | Homo sapiens | 2 | ALA4402604 | single protein format | Scientific Literature | |
14. | ALA4406332 | B | Binding affinity to recombinant PI5P4Kbeta (unknown origin) assessed as protein-labeling at 10 uM incubated for 2 hrs by mass spectrometry | Homo sapiens | 2 | ALA4402604 | single protein format | Scientific Literature | |
15. | ALA4406349 | B | Binding affinity to human PI5P4IKgamma | Homo sapiens | 4 | ALA4402604 | single protein format | Scientific Literature | |
16. | ALA5045820 | B | Inhibition of PI5P4Kgamma (unknown origin) at 1 uM by KINOMEscan analysis | Homo sapiens | 3 | ALA5042546 | single protein format | Scientific Literature | |
17. | ALA5260676 | B | Inhibition of PI5P4Kalpha (unknown origin) | Homo sapiens | 2 | ALA5257158 | single protein format | Scientific Literature |