| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4355751 | A | Apparent permeability in pig LLC-PK1 cells transfected with MDR1 | Sus scrofa | 25 | cell-based format | Scientific Literature | ||
| 2. | ALA4355754 | B | Inhibition of recombinant human OGA | Homo sapiens | 48 | single protein format | Scientific Literature | ||
| 3. | ALA4355755 | B | Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISA | Rattus norvegicus | 25 | cell-based format | Scientific Literature | ||
| 4. | ALA4355756 | B | Inhibition of human beta hexosaminidase assessed as inhibitory constant using 4-methylumbelliferyl N-acetyl-beta-D-glucosaminide dihydrate as substrate measured every 60 sec for 45 mins by fluorescence spectrophotometry | Homo sapiens | 41 | single protein format | Scientific Literature | ||
| 5. | ALA4355758 | A | AUCN in Wistar Han rat at 10 mg/kg, po | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 6. | ALA4355760 | A | Clearance in Wistar Han rat at 2 mg/kg, iv | Rattus norvegicus | 18 | organism-based format | Scientific Literature | ||
| 7. | ALA4355762 | A | Half life in Wistar Han rat at 2 mg/kg, iv | Rattus norvegicus | 17 | organism-based format | Scientific Literature | ||
| 8. | ALA4355764 | A | Volume of distribution at steady state in Wistar Han rat at 2 mg/kg, iv or 10 mg/kg, po | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 9. | ALA4355767 | A | Oral bioavailability in Wistar Han rat at 10 mg/kg | Rattus norvegicus | 7 | organism-based format | Scientific Literature | ||
| 10. | ALA4355799 | B | Displacement of MK-0499 from human ERG | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 11. | ALA4355800 | B | Inhibition of Nav1.5 (unknown origin) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 12. | ALA4355801 | B | Inhibition of Cav1.2 (unknown origin) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 13. | ALA4355802 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 14. | ALA4355803 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 15. | ALA4355804 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 16. | ALA4355805 | B | Activation of PXR (unknown origin) assessed as CYP3A4 induction | Homo sapiens | 11 | single protein format | Scientific Literature |
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