| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4332153 | B | Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-based luciferase reporter gene assay | Homo sapiens | 35 | cell-based format | Scientific Literature | ||
| 2. | ALA4332154 | B | Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-based luciferase reporter gene assay | Homo sapiens | 35 | cell-based format | Scientific Literature | ||
| 3. | ALA4332155 | A | Transactivation of PXR (unknown origin) assessed as CYP450 induction at 10 uM relative to 10 uM rifampicin | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 4. | ALA4332156 | A | Transactivation of PXR (unknown origin) assessed as increase in CYP3A4 mRNA expression at 10 uM relative to 10 uM rifampicin | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 5. | ALA4332157 | B | Antagonist activity at PPARgamma (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4332158 | B | Agonist activity at recombinant human PPARalpha after overnight incubation by cell-based luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA4332159 | B | Agonist activity at recombinant human PPARdelta after overnight incubation by cell-based luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA4332160 | B | Agonist activity at PPARgamma (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4332161 | B | Antagonist activity at mouse PPARalpha | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4332162 | B | Antagonist activity at mouse PPARdelta | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4332163 | B | Antagonist activity at mouse PPARgamma | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4332164 | B | Antagonist activity at ERbeta receptor (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4332165 | B | Antagonist activity at glucocorticoid receptor (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4332166 | B | Antagonist activity at thyroid hormone receptor (unknown origin) | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 15. | ALA4332167 | B | Antagonist activity at retinoid X receptor (unknown origin) | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 16. | ALA4332168 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4332169 | A | Cytotoxicity against CHO cells assessed as effect on cell viability | Cricetulus griseus | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4332170 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4332171 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4332172 | A | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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