# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4364841 | B | Inhibition of Plasmodium falciparum 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate in presence of beta2 inhibitor WLW-VS | Plasmodium falciparum | 27 | ALA4364250 | assay format | Scientific Literature | |
2. | ALA4364842 | A | Inhibition of human beta5 20S constitutive proteasome using suc-LLVY-AMC as substrate | Homo sapiens | 27 | ALA4364250 | single protein format | Scientific Literature | |
3. | ALA4364843 | A | Inhibition of human beta5 20S immunoproteasome using Ac-ANW-AMC as substrate | Homo sapiens | 27 | ALA4364250 | single protein format | Scientific Literature | |
4. | ALA4364844 | F | Antimalarial activity against erythrocytic stage of Plasmodium falciparum 3D7 measured after 72 hrs by SYBR green dye based fluorescence assay | Plasmodium falciparum | 27 | ALA4364250 | organism-based format | Scientific Literature | |
5. | ALA4364845 | T | Selectivity ratio of IC50 for human beta5 20S constitutive proteasome to IC50 for Plasmodium falciparum 20S proteasome beta5 subunit | 24 | ALA4364250 | assay format | Scientific Literature | ||
6. | ALA4364846 | T | Selectivity ratio of IC50 for human beta5 20S immunoproteasome to IC50 for Plasmodium falciparum 20S proteasome beta5 subunit | 24 | ALA4364250 | assay format | Scientific Literature | ||
7. | ALA4364850 | A | Cytotoxicity against human HepG2 cells | Homo sapiens | 24 | ALA4364250 | cell-based format | Scientific Literature | |
8. | ALA4364851 | A | Cytotoxicity against human KARPAS1106P cells | Homo sapiens | 24 | ALA4364250 | cell-based format | Scientific Literature |