# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4388469 | B | Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as substrate measured at 30 secs interval for 5 mins by fluorescence intensity assay | Homo sapiens | 27 | ALA4387717 | cell-based format | Scientific Literature | |
2. | ALA4388470 | A | Inhibition of recombinant bovine enterokinase activated N-terminal His-tagged recombinant human KLK1 (19 to 262 residues) expressed in baculovirus infected Sf9 insect cells using 3',6'-bis(prolylphenylalanylarginylamino)3H-spiro(2-benzofuran-1,9'-xanthen)-3-one;TFA as substrate measured at 30 secs interval for 5 mins by fluorescence intensity assay | Homo sapiens | 27 | ALA4387717 | cell-based format | Scientific Literature | |
3. | ALA4424180 | B | Inhibition of recombinant human FLAG-tagged KLK5 expressed in baculovirus infected sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as substrate measured every 30 secs intervals for 5 mins by Rhodamine110 dye-based fluorescence assay | Homo sapiens | 15 | ALA4422656 | cell-based format | Scientific Literature | |
4. | ALA4424181 | B | Inhibition of recombinant human N-terminal his-tagged KLK1 (19 to 262 residues) expressed in baculovirus infected sf9 insect cells using R110 labelled GSK3162232A as substrate measured every 30 secs intervals for 5 mins by Rhodamine110 dye-based fluorescence assay | Homo sapiens | 15 | ALA4422656 | cell-based format | Scientific Literature | |
5. | ALA4424183 | B | Selectivity ratio of IC50 for recombinant human N-terminal his-tagged KLK1 (19 to 262 residues) to IC50 for recombinant human FLAG-tagged KLK5 | Homo sapiens | 3 | ALA4422656 | assay format | Scientific Literature |