| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4343178 | B | Inhibition of recombinant human C-terminal GST/His-tagged HDAC3 (1 to 428 residues) co-expressed with human N-terminal GST-tagged NCOR2 (395 to 489 residues) in baculovirus infected Sf9 cells using Boc-Lys(Ac)-AMC as substrate preincubated for 15 mins followed by substrate addition and measured after 60 mins by fluorometric method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 2. | ALA4343179 | F | Growth inhibition of human THP1 cells incubated for 72 hrs by trypan blue assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA4343180 | B | Inhibition of GST-tagged BRD4 bromodomain 1/2 (unknown origin) at 10 uM incubated for 3 hrs by fluorescence based assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA4725765 | B | Inhibition of HDAC1 (unknown origin) | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 5. | ALA4725766 | B | Inhibition of BRD4 (unknown origin) | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 6. | ALA4770956 | B | Inhibition of recombinant human HDAC1 using Z-(Ac)Lys-AMC as substrate after 90 mins by fluorescence based micro plate assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 7. | ALA4770993 | B | Inhibition of HDAC2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4770994 | B | Inhibition of HDAC3 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4770995 | B | Inhibition of BRD4 (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4819310 | B | Inhibition of C-terminal His-tagged human HDAC3 (1 to 428 residues)/N-terminal GST tagged human NCOR2 (395 to 489) expressed in baculovirus expression system using Boc-Lys(Ac)-AMC as substrate preincubated for 15 mins followed by substrate addition and measured after 60 mins by fluorescence method | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4819311 | F | Antiproliferative activity against human THP1 incubated for 72 hrs by Trypan Blue reagent based assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA5096335 | B | Inhibition of human HDAC3 using Boc-Lys(Ac)-AMC as substrate by fluorescence based assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 13. | ALA5096336 | B | Inhibition of GST-tagged BRD4 (unknown origin) at 10 uM by HTRF assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA5234196 | B | Inhibition of human HDAC1 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assay | Homo sapiens | 11 | subcellular format | Scientific Literature | ||
| 15. | ALA5234197 | B | Inhibition of human HDAC2 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assay | Homo sapiens | 11 | subcellular format | Scientific Literature | ||
| 16. | ALA5234198 | B | Inhibition of human HDAC3 using human HeLa cell nuclear extract at 1 uM measured after 60 mins by fluorescence assay | Homo sapiens | 11 | subcellular format | Scientific Literature | ||
| 17. | ALA5245804 | B | Inhibition of human full length BRD4 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA5245805 | B | Inhibition of human full length BRD4 at 10 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |
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