| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4406333 | B | Inhibition of GST-tagged recombinant PI5P4Kalpha (unknown origin) incubated for 1 hr in presence of DPPS and PI5P by ADP-Glo assay | Homo sapiens | 24 | ALA4402604 | single protein format | Scientific Literature | |
| 2. | ALA4406334 | B | Inhibition of GST-tagged recombinant PI5P4Kbeta (unknown origin) incubated for 1 hr in presence of DPPS and PI5P by ADP-Glo assay | Homo sapiens | 24 | ALA4402604 | single protein format | Scientific Literature | |
| 3. | ALA4406335 | P | Lipophilicity, logD of the compound | 24 | ALA4402604 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA4406336 | B | Induction of stabilization of PI5P4Kalpha in HEK293T cells at 1 to 15 uM incubated for 1 hr at 40 to 67 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 4 | ALA4402604 | cell-based format | Scientific Literature | |
| 5. | ALA4406337 | B | Induction of stabilization of PI5P4Kbeta in HEK293T cells at 1 to 15 uM incubated for 1 hr at 40 to 67 degC by Western blot analysis based isothermal CETSA method | Homo sapiens | 3 | ALA4402604 | cell-based format | Scientific Literature | |
| 6. | ALA4406338 | A | Permeability of the compound by PAMPA method | 3 | ALA4402604 | assay format | Scientific Literature | ||
| 7. | ALA4406339 | A | Stability in rat liver microsomes at 1 uM in presence of NADPH regeneration system incubated for 15 mins by LC-MS analysis | Rattus norvegicus | 4 | ALA4402604 | microsome format | Scientific Literature | |
| 8. | ALA4406345 | B | Inhibition of human ACVR2B expressed in baculovirus expression system | Homo sapiens | 3 | ALA4402604 | assay format | Scientific Literature | |
| 9. | ALA4406346 | B | Inhibition of human TGFBR2 expressed in baculovirus expression system | Homo sapiens | 3 | ALA4402604 | assay format | Scientific Literature | |
| 10. | ALA4406349 | B | Binding affinity to human PI5P4IKgamma | Homo sapiens | 4 | ALA4402604 | single protein format | Scientific Literature | |
| 11. | ALA4406350 | B | Inhibition of human ACVR2A expressed in baculovirus expression system | Homo sapiens | 1 | ALA4402604 | assay format | Scientific Literature | |
| 12. | ALA5045820 | B | Inhibition of PI5P4Kgamma (unknown origin) at 1 uM by KINOMEscan analysis | Homo sapiens | 3 | ALA5042546 | single protein format | Scientific Literature | |
| 13. | ALA5045821 | B | Inhibition of PI5P4Kalpha (unknown origin) by bioluminescent assay | Homo sapiens | 1 | ALA5042546 | single protein format | Scientific Literature | |
| 14. | ALA5045822 | B | Inhibition of PI5P4Kbeta (unknown origin) by fluorescence polarization assay | Homo sapiens | 1 | ALA5042546 | single protein format | Scientific Literature |
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