| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4384529 | F | Growth inhibition of human KB cells after 48 hrs by SRB assay | Homo sapiens | 23 | ALA4382249 | cell-based format | Scientific Literature | |
| 2. | ALA4384530 | F | Growth inhibition of human A549 cells after 48 hrs by SRB assay | Homo sapiens | 23 | ALA4382249 | cell-based format | Scientific Literature | |
| 3. | ALA4384531 | F | Growth inhibition of human MKN45 cells after 48 hrs by SRB assay | Homo sapiens | 23 | ALA4382249 | cell-based format | Scientific Literature | |
| 4. | ALA4384532 | F | Growth inhibition of human KB-VIN10 cells after 48 hrs by SRB assay | Homo sapiens | 3 | ALA4382249 | assay format | Scientific Literature | |
| 5. | ALA4384533 | F | Growth inhibition of human KB-S15 cells after 48 hrs by SRB assay | Homo sapiens | 3 | ALA4382249 | assay format | Scientific Literature | |
| 6. | ALA4384534 | F | Growth inhibition of human KB-7d cells after 48 hrs by SRB assay | Homo sapiens | 3 | ALA4382249 | assay format | Scientific Literature | |
| 7. | ALA4384535 | B | Inhibition of human HDAC6 in human A549 cells assessed as increase in acetylated alpha-tubulin level at 0.6 to 2.5 uM after 6 hrs by Western blot analysis | Homo sapiens | 1 | ALA4382249 | cell-based format | Scientific Literature | |
| 8. | ALA4384536 | B | Inhibition of bovine brain tubulin polymerization measured every 30 secs for 30 mins by turbidimetric assay | Bos taurus | 24 | ALA4382249 | assay format | Scientific Literature | |
| 9. | ALA4384537 | B | Displacement of [3H]-colchicine from bovine brain tubulin at 1 uM by scintillation proximity assay relative to control | Bos taurus | 24 | ALA4382249 | assay format | Scientific Literature | |
| 10. | ALA4384538 | B | Displacement of [3H]-colchicine from bovine brain tubulin at 5 uM by scintillation proximity assay relative to control | Bos taurus | 24 | ALA4382249 | assay format | Scientific Literature | |
| 11. | ALA4384539 | B | Inhibition of human HDAC1 using RHKKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 12. | ALA4384540 | B | Inhibition of human HDAC2 using RHKKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 13. | ALA4384541 | B | Inhibition of human HDAC3 using RHKKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 14. | ALA4384542 | B | Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 15. | ALA4384543 | B | Inhibition of human HDAC6 using RHKKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 16. | ALA4384544 | B | Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 17. | ALA4384545 | B | Inhibition of human HDAC8 using RHKAcKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 18. | ALA4384546 | B | Inhibition of human HDAC9 using Boc-Lys(trifluoroacetyl)-AMC as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 19. | ALA4384547 | B | Inhibition of human HDAC10 using RHKKAc as substrate by fluorescence assay | Homo sapiens | 3 | ALA4382249 | single protein format | Scientific Literature | |
| 20. | ALA4384548 | F | Antitumor activity against human A549 cells xenografted in Balb/c nude mouse assessed as tumor growth inhibition at 50 mg/kg, ip daily measured up to 18 days relative to control | Homo sapiens | 1 | ALA4382249 | organism-based format | Scientific Literature |
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