| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4425846 | Binding | Inhibition of recombinant His-tagged BRD4 bromodomain1 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 2. | ALA4425847 | Binding | Inhibition of recombinant His-tagged BRD4 bromodomain2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 3. | ALA4425848 | Binding | Displacement of biotinylated JQ1 analog from recombinant His-tagged CBP (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 4. | ALA4425849 | Binding | Displacement of biotinylated JQ1 analog from recombinant His-tagged BRPF1 (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 5. | ALA4425850 | Binding | Displacement of biotinylated JQ1 analog from recombinant His-tagged BRD9 (unknown origin) incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 6. | ALA4425851 | Binding | Inhibition of recombinant His-tagged TAF1 isoform-1 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 7. | ALA4425852 | Binding | Inhibition of recombinant His-tagged TAF1 isoform-2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 8. | ALA4425853 | Binding | Inhibition of recombinant His-tagged CECR2 (unknown origin) using biotinylated ligand incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA4425103 | single protein format | Scientific Literature | |
| 9. | ALA4425856 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged BRD4 bromodomain1 to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 10. | ALA4425857 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged BRD4 bromodomain2 to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 11. | ALA4425858 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged CBP (unknown origin) to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 12. | ALA4425859 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged BRPF1 (unknown origin) to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 13. | ALA4425860 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged TAF1 isoform-1 (unknown origin) to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 14. | ALA4425861 | Binding | Selectivity index, ratio of IC50 for recombinant His-tagged TAF2 isoform-1 (unknown origin) to IC50 for recombinant His-tagged CECR2 (unknown origin) | Homo sapiens | 1 | ALA4425103 | assay format | Scientific Literature | |
| 15. | ALA4425865 | Binding | Binding affinity to wild type CECR2 (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | ALA4425103 | single protein format | Scientific Literature | |
| 16. | ALA4425866 | Binding | Binding affinity to CECR2 Y520I mutant (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | ALA4425103 | single protein format | Scientific Literature | |
| 17. | ALA4425867 | Binding | Binding affinity to CECR2 M506I mutant (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO red dye based differential scanning fluorimetry | Homo sapiens | 2 | ALA4425103 | single protein format | Scientific Literature | |
| 18. | ALA4425868 | Binding | Binding affinity to human partial length CECR2 expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 4 | ALA4425103 | assay format | Scientific Literature |
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