| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4398063 | Binding | Inhibition of PRMT4 (unknown origin) using histone H3 (21 to 44 residues) as substrate measured after 60 mins in presence of SAM by AlphaLisa assay | Homo sapiens | 44 | ALA4396888 | single protein format | Scientific Literature | |
| 2. | ALA4398064 | Binding | Inhibition of PRMT1 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 2 | ALA4396888 | single protein format | Scientific Literature | |
| 3. | ALA4398065 | Binding | Inhibition of PRMT6 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 2 | ALA4396888 | single protein format | Scientific Literature | |
| 4. | ALA4398066 | Binding | Selectivity ratio of IC50 for PRMT1 (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 2 | ALA4396888 | assay format | Scientific Literature | |
| 5. | ALA4398067 | Binding | Selectivity ratio of IC50 for PRMT6 (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 2 | ALA4396888 | assay format | Scientific Literature | |
| 6. | ALA4398068 | Binding | Inhibition of recombinant full-length human PRMT7 expressed in Sf9 insect cells using Ac-KKDGKKRKRSRKESYK-biotin as substrate measured after 30 mins in presence of SAM by topcount scintillation counting method | Homo sapiens | 1 | ALA4396888 | cell-based format | Scientific Literature | |
| 7. | ALA4398069 | Binding | Inhibition of PRMT3 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 8. | ALA4398070 | Binding | Inhibition of PRMT8 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 9. | ALA4398071 | Binding | Inhibition of PRMT5 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 10. | ALA4398072 | Binding | Selectivity ratio of IC50 for PRMT3 (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 1 | ALA4396888 | assay format | Scientific Literature | |
| 11. | ALA4398073 | Binding | Selectivity ratio of IC50 for PRMT8 (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 1 | ALA4396888 | assay format | Scientific Literature | |
| 12. | ALA4398074 | Binding | Selectivity ratio of IC50 for PRMT5 (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 1 | ALA4396888 | assay format | Scientific Literature | |
| 13. | ALA4398075 | Binding | Selectivity ratio of IC50 for recombinant full-length human PRMT7 expressed in Sf9 insect cells (unknown origin) to IC50 for PRMT4 (unknown origin) | Homo sapiens | 1 | ALA4396888 | cell-based format | Scientific Literature | |
| 14. | ALA4398076 | Binding | Inhibition of EZH2 (unknown origin) up to 50 uM preincubated for 10 mins followed by peptide substrate addition and measured after 4 hrs in presence of SAM by HTRF assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 15. | ALA4398077 | Binding | Inhibition of MLL1 (unknown origin) up to 50 uM preincubated for 10 mins followed by peptide substrate addition and measured after 4 hrs in presence of SAM by HTRF assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 16. | ALA4398078 | Binding | Inhibition of NSD2 (unknown origin) up to 50 uM preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 17. | ALA4398079 | Binding | Inhibition of SMYD3 (unknown origin) up to 50 uM preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 18. | ALA4398080 | Binding | Inhibition of DOT1L (unknown origin) up to 50 uM preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 19. | ALA4398081 | Binding | Inhibition of G9a (unknown origin) up to 50 uM preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLisa assay | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature | |
| 20. | ALA4398082 | Binding | Inhibition of SETD2 (unknown origin) up to 50 uM | Homo sapiens | 1 | ALA4396888 | single protein format | Scientific Literature |
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