| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4411099 | B | Inhibition of human GRK5 using tubulin as substrate measured after 0 mins by [gamma-32P]-ATP assay | Homo sapiens | 7 | ALA4406919 | single protein format | Scientific Literature | |
| 2. | ALA4411100 | B | Inhibition of human GRK5 using tubulin as substrate measured after 30 mins by [gamma-32P]-ATP assay | Homo sapiens | 6 | ALA4406919 | single protein format | Scientific Literature | |
| 3. | ALA4411101 | B | Inhibition of human GRK5 using tubulin as substrate measured after 60 mins by [gamma-32P]-ATP assay | Homo sapiens | 6 | ALA4406919 | single protein format | Scientific Literature | |
| 4. | ALA4411102 | B | Inhibition of human GRK5 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Homo sapiens | 12 | ALA4406919 | single protein format | Scientific Literature | |
| 5. | ALA4411103 | B | Inhibition of bovine GRK1 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 6 | ALA4406919 | single protein format | Scientific Literature | |
| 6. | ALA4411104 | B | Inhibition of bovine GRK2 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 16 | ALA4406919 | single protein format | Scientific Literature | |
| 7. | ALA4411105 | B | Inhibition of bovine GRK6 using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 12 | ALA4406919 | assay format | Scientific Literature | |
| 8. | ALA4411106 | B | Inhibition of bovine GRK5 C474S mutant using tubulin as substrate measured after 4 hrs by [gamma-32P]-ATP assay | Bos taurus | 5 | ALA4406919 | single protein format | Scientific Literature | |
| 9. | ALA4411107 | B | Inhibition of human GRK5 using light activated ROS as substrate measured after 0 mins to 4 hrs by [gamma-32P]-ATP assay | Homo sapiens | 1 | ALA4406919 | single protein format | Scientific Literature | |
| 10. | ALA4411108 | B | Selectivity index, ratio of IC50 for bovine GRK2 to IC50 for human GRK5 | 16 | ALA4406919 | assay format | Scientific Literature | ||
| 11. | ALA4411109 | B | Covalent inhibition of human GRK5 assessed as adduct appearance incubated for 3 hrs by intact protein mass spectroscopy | Homo sapiens | 11 | ALA4406919 | single protein format | Scientific Literature |
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