| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4394427 | F | Antiproliferative activity against human PC3 cells measured after 72 hrs by celltiter-glo assay | Homo sapiens | 7 | ALA4393668 | cell-based format | Scientific Literature | |
| 2. | ALA4394428 | F | Antiproliferative activity against human DU145 cells measured after 72 hrs by celltiter-glo assay | Homo sapiens | 7 | ALA4393668 | cell-based format | Scientific Literature | |
| 3. | ALA4394429 | F | Antiproliferative activity against human C4-2B cells measured after 96 hrs by celltiter-glo assay | Homo sapiens | 7 | ALA4393668 | cell-based format | Scientific Literature | |
| 4. | ALA4394430 | B | Inverse agonist activity at Gal4-fused RORgamma LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay | Homo sapiens | 26 | ALA4393668 | cell-based format | Scientific Literature | |
| 5. | ALA4394432 | B | Binding affinity to human N-terminal His6-tagged RORgamma (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) assessed as change in melting temperature at 200 uM by SYPRO orange-dye based fluorescence assay | Homo sapiens | 26 | ALA4393668 | assay format | Scientific Literature | |
| 6. | ALA4394433 | B | Inverse agonist activity at Gal4-fused RORalpha LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay | Homo sapiens | 6 | ALA4393668 | cell-based format | Scientific Literature | |
| 7. | ALA4394434 | B | Inverse agonist activity at Gal4-fused RORbeta LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay | Homo sapiens | 6 | ALA4393668 | cell-based format | Scientific Literature | |
| 8. | ALA4394435 | B | Inverse agonist activity at Gal4-fused LXRalpha LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay | Homo sapiens | 5 | ALA4393668 | cell-based format | Scientific Literature | |
| 9. | ALA4394436 | B | Inverse agonist activity at Gal4-fused FXR LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay | Homo sapiens | 5 | ALA4393668 | cell-based format | Scientific Literature | |
| 10. | ALA4394437 | B | Inverse agonist activity at Gal4-fused RORalpha LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay relative to control | Homo sapiens | 3 | ALA4393668 | cell-based format | Scientific Literature | |
| 11. | ALA4394440 | B | Inverse agonist activity at Gal4-fused FXR LBD (unknown origin) expressed in 293T cells measured after 24 hrs by dual-luciferase reporter gene assay relative to control | Homo sapiens | 1 | ALA4393668 | cell-based format | Scientific Literature | |
| 12. | ALA4394441 | B | Inverse agonist activity at human N-terminal His6-tagged RORgamma (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition of biotinylated co-activator SRC1-4 peptide recruitment by alphascreen assay | Homo sapiens | 5 | ALA4393668 | assay format | Scientific Literature | |
| 13. | ALA4394443 | F | Antiproliferative activity against human LNCAP cells measured after 96 hrs by celltiter-glo assay | Homo sapiens | 7 | ALA4393668 | cell-based format | Scientific Literature | |
| 14. | ALA4394444 | F | Antiproliferative activity against human 22Rv1 cells measured after 96 hrs by celltiter-glo assay | Homo sapiens | 7 | ALA4393668 | cell-based format | Scientific Literature |
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